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PROTAC ER Degrader-4

PROTAC ER Degrader-4 Structure
PROTAC ER Degrader-4 structure
CAS No.
2361114-15-8
Chemical Name:
PROTAC ER Degrader-4
Synonyms
PROTAC ER Degrader-4
CBNumber:
CB28054603
Molecular Formula:
C53H67F3N6O8S
Molecular Weight:
1005.19
MDL Number:
MFCD34469813
MOL File:
Mol file
Last updated:2023-02-23 14:24:06
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PROTAC ER Degrader-4 Properties

Boiling point 1038.9±65.0 °C(Predicted)
Density 1.254±0.06 g/cm3(Predicted)
pka 13.54±0.46(Predicted)

PROTAC ER Degrader-4 Chemical Properties,Uses,Production

Biological Activity

PROTAC ER Degrader-4 is a von Hippel-Lindau-based PROATC estrogen receptor (ER) degrader, binding to ER with an IC50 of 0.8 nM. PROTAC ER Degrader-4 induces ER degradation in MCF-7 cells with an IC50 of 0.3 nM[1]. PROTAC ER Degrader-4 shows equal to 100% ER degradation at 0.3 μM in the MCF-7 ER degradation cellular assay[1].

References

[1]. Bin Yang, et al. Compounds and their use in treating cancer. WO2019123367A1.

PROTAC ER Degrader-4 Preparation Products And Raw materials

Raw materials

Preparation Products

PROTAC ER Degrader-4 Suppliers

Global( 5)Suppliers
Supplier Tel Email Country ProdList Advantage
TargetMol Chemicals Inc. 		+1-781-999-5354 +1-00000000000 marketing@targetmol.com United States 19892 58
Sichuan Wei Keqi Biological Technology Co., Ltd. 028-81700200 18116577057 3003855609@qq.com China 7892 56
Shanghai Chaolan Chemical Technology Center QQ:65489617 15618227136 info@SuperLan-chem.com China 9833 58
Jilin Province Woda Biotechnology Co., Ltd. 13504435624 1927928688@qq.com China 1360 58
Changzhou Bojia Biomedical Technology Co., Ltd. 2122619822 czbjpharma@126.com China 18488 58
Supplier Advantage
TargetMol Chemicals Inc. 		58
Sichuan Wei Keqi Biological Technology Co., Ltd. 56
Shanghai Chaolan Chemical Technology Center 58
Jilin Province Woda Biotechnology Co., Ltd. 58
Changzhou Bojia Biomedical Technology Co., Ltd. 58

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PROTAC ER Degrader-4 2361114-15-8