Meptazinol hydrochloride
- CAS No.
- 59263-76-2
- Chemical Name:
- Meptazinol hydrochloride
- Synonyms
- Meptazinol hcl;Meptazinol-d3 HCl;Meptazinol hydrochlo;WY-22811 hydrochloride;IL-22811 hydrochloride;MEPTAZINOL HYDROCHLORIDE;Meptazinol-d3 hydrochloride;Meptazinol hydrochloride USP/EP/BP;IL-22811 HYDROCHLORIDE;WY-22811 HYDROCHLORIDE;3-(3-ethyl-1-methyl-3-azepanyl)phenol hydrochloride
- CBNumber:
- CB4843649
- Molecular Formula:
- C15H24ClNO
- Molecular Weight:
- 269.81
- MDL Number:
- MFCD00941476
- MOL File:
- 59263-76-2.mol
| Melting point | 250-252°C |
|---|---|
| storage temp. | Inert atmosphere,2-8°C |
| solubility | H2O: >10mg/mL |
| form | powder |
| color | white to off-white |
| Stability | Hygroscopic |
| InChIKey | MPJUSISYVXABBH-UHFFFAOYSA-N |
| FDA UNII | T62FQ4ZCPA |
SAFETY
Risk and Safety Statements
| Symbol(GHS) |  GHS07 |
|---|---|
| Signal word | Warning |
| Hazard statements | H302 |
| Precautionary statements | P264-P270-P301+P312+P330-P501 |
| Hazard Codes | Xn |
| Risk Statements | 22 |
| WGK Germany | 1 |
| RTECS | SL4250000 |
Meptazinol hydrochloride price More Price(42)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Sigma-Aldrich | M2824 | Meptazinol hydrochloride | 59263-76-2 | 10mg | $91.6 | 2024-03-01 | Buy |
| Sigma-Aldrich | BP583 | Meptazinol hydrochloride British Pharmacopoeia (BP) Reference Standard | 59263-76-2 | 100MG | $229 | 2024-03-01 | Buy |
| Sigma-Aldrich | M2824 | Meptazinol hydrochloride | 59263-76-2 | 50mg | $314 | 2022-05-15 | Buy |
| Tocris | 3636 | Meptazinol hydrochloride ≥99%(HPLC) | 59263-76-2 | 50 | $331 | 2021-12-16 | Buy |
| Tocris | 3636 | Meptazinol hydrochloride ≥99%(HPLC) | 59263-76-2 | 10 | $83 | 2021-12-16 | Buy |
Meptazinol hydrochloride Chemical Properties,Uses,Production
Description
Meptazinol hydrochloride is an injectable narcotic analgesic with antagonist properties; it is similar in potency to meperidine. Meptazinol appears to have a low propensity toward respiratory depression and other opiate-like side effects, possibly due to selective interaction with the mu-1 receptor. Also somewhat unique for an analgesic, it interacts with central cholinergic receptors. An oral form of meptazinol is under development.
Chemical Properties
White Solid
Originator
Wyeth (United Kingdom)
Uses
Mixed opioid agonist-antagonist. Analgesic (narcotic).
Uses
Analgesic;Opiate receptor agonist
brand name
MEPTID
Biological Activity
Centrally active opioid analgesic. Partial agonist at the μ 1 opioid receptor. Also shown to inhibit acetylcholinesterase.
Biochem/physiol Actions
Meptazinol entered the human pharmaceutical market as a racemic mixture in the 1980s for use as an analgesic. Its pharmacology is not completely understood; however, its analgesic properties are mostly due to its partial agonism at the mu1 opioid receptor. Due to its partial agonism, Meptazinol antagonizes morphine dependence in vivo. Its advantage over other opiates is its reduced capacity to cause addition and respiratory depression, also due to its intrinsic activity as a partial agonist. Meptazinol has been found to have additional activity as an acetylcholinesterase (AChE) inhibitor, particularly in its (-) enantiomeric form, which may partially explain its analgesic properties. AChE inhibitors are used to treat Alzheimer′s disease, providing additional interest in this compound.
Meptazinol hydrochloride Preparation Products And Raw materials
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| Xiamen Wonderful Bio Technology Co., Ltd. | +8613043004613 | Sara@xmwonderfulbio.com | China | 305 | 58 |
| Henan Tianfu Chemical Co.,Ltd. | +86-0371-55170693 +86-19937530512 | info@tianfuchem.com | China | 21695 | 55 |
| Hangzhou FandaChem Co.,Ltd. | 008657128800458; +8615858145714 | fandachem@gmail.com | China | 9348 | 55 |
| Shanghai Zheyan Biotech Co., Ltd. | 18017610038 | zheyansh@163.com | CHINA | 3620 | 58 |
| career henan chemical co | +86-0371-86658258 | sales@coreychem.com | China | 29914 | 58 |
| Chongqing Chemdad Co., Ltd | +86-023-61398051 +8613650506873 | sales@chemdad.com | China | 39916 | 58 |
| CONIER CHEM AND PHARMA LIMITED | +8618523575427 | sales@conier.com | China | 47465 | 58 |
| Shaanxi Dideu Medichem Co. Ltd | +86-29-87569265 +86-18612256290 | 1056@dideu.com | China | 3683 | 58 |
| SIMAGCHEM CORP | +86-13806087780 | sale@simagchem.com | China | 17367 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354 +1-00000000000 | marketing@targetmol.com | United States | 19892 | 58 |
View Lastest Price from Meptazinol hydrochloride manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
 |
2024-01-18 | Meptazinol HCl
59263-76-2
|
US $120.00 / KG | 1250KG | 99.8% | 330T | Xiamen Wonderful Bio Technology Co., Ltd. | |
 |
2021-07-20 | Meptazinol hydrochloride
59263-76-2
|
US $1.00-1.00 / Kg/Bag | 1g | 99% | 50tons | Shaanxi Dideu Medichem Co. Ltd | |
 |
2021-06-11 | Meptazinol hydrochloride USP/EP/BP
59263-76-2
|
US $1.10 / g | 1g | 99.9% | 100 Tons Min | Dideu Industries Group Limited |
-
- Meptazinol HCl
59263-76-2
- US $120.00 / KG
- 99.8%
- Xiamen Wonderful Bio Technology Co., Ltd.
-
- Meptazinol hydrochloride
59263-76-2
- US $1.00-1.00 / Kg/Bag
- 99%
- Shaanxi Dideu Medichem Co. Ltd
-
- Meptazinol hydrochloride USP/EP/BP
59263-76-2
- US $1.10 / g
- 99.9%
- Dideu Industries Group Limited