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Fabesetron

CAS No.
129300-27-2
Chemical Name:
Fabesetron
Synonyms
Fabesetron;Fabesetron [INN];FK1052 free base;Pyrido[1,2-a]indol-6(7H)-one, 8,9-dihydro-10-methyl-7-[(4-methyl-1H-imidazol-5-yl)methyl]-, (7R)-
CBNumber:
CB61178694
Molecular Formula:
C18H19N3O
Molecular Weight:
293.36
MDL Number:
MFCD00891468
MOL File:
129300-27-2.mol
Last updated:2023-05-04 17:34:32

Fabesetron Properties

FDA UNII QU72HVX338

Fabesetron Chemical Properties,Uses,Production

Definition

ChEBI: Fabesetron is an organic heterotricyclic compound that is 8,9-dihydropyrido[1,2-a]indol-6(7H)-one substituted by a (5-methyl-1H-imidazol-4-yl)methyl group at position 7R and a methyl group at position 10. It is a dual 5-HT3 and 5-HT4 receptors antagonist whose clinical development was terminated in phase II. It was being developed for the treatment of chemotherapy-induced emesis and irritable bowel syndrome. It has a role as an antiemetic and a serotonergic antagonist. It is a member of imidazoles and an organic heterotricyclic compound.

Fabesetron Preparation Products And Raw materials

Raw materials

Preparation Products

Fabesetron Suppliers

Global( 5)Suppliers
Supplier Tel Email Country ProdList Advantage
Beijing Jin Ming Biotechnology Co., Ltd. 010-60605840 15801484223 psaitong@jm-bio.com China 29834 58
Changzhou Bojia Biomedical Technology Co., Ltd. 2122619822 czbjpharma@126.com China 18488 58
Fabesetron Fabesetron [INN] Pyrido[1,2-a]indol-6(7H)-one, 8,9-dihydro-10-methyl-7-[(4-methyl-1H-imidazol-5-yl)methyl]-, (7R)- FK1052 free base 129300-27-2