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主营产品:1)以含氟药物分子砌块和手性药物分子砌块为特色的高品质的药物分子砌块以及原创新药关键砌块;(2)原创新药关键砌块的工艺开发、中试、商业化生产和销售。

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    南京优氟医药科技有限公司

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  • 产品总数:2358
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  • 国籍:中国
  •       南京优氟医药科技有限公司由归国科学家博士团队于2018年创建,致力于为全球原创新药研发机构和生产企业提供有特色的医药化学产品和专业的新药研发技术服务。公司创始团队在原创新药研发领域拥有丰富经验,获得“江苏省双创人才”、“南京市高层次创业人才”、“江苏省产业教授”等荣誉头衔。 依托公司在药物化学、有机氟化学、工艺化学、手性化学、多步骤有机合成化学、药物分析化学等领域的核心技术优势,公司的核心业务包括:(1)以含氟药物分子砌块和手性药物分子砌块为特色的药物分子砌块的设计、研发、制造、销售;(2)原创新药关键砌块的工艺开发、中试、商业化生产和销售。公司自成立以来快速发展,与国内外原创新药领域内的制药龙头企业、CRO头部企业、主流商贸企业和科研院所形成密切的合作关系,并于2019年获评“江苏省技术先进型服务企业”,2020年获评“国家高新技术企业”。
英文名称 中文名称 CAS号 操作
tert-butyl (R)-4-(difluoromethyl)-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide (R)-4-(二氟甲基)-1,2,3-噁噻唑烷-3-羧酸叔丁酯2,2-二氧化物 3007737-61-0 详细
(3S,5R)-5-(trifluoromethyl)pyrrolidin-3-ol 详细
tert-butyl (2R,4R)-4-hydroxy-2-methylpyrrolidine-1-carboxylate (2R,4R)-N-Boc-4-羟基-2-甲基吡咯烷 114676-93-6 详细
(3S,5S)-5-methylpyrrolidin-3-ol (3S,5S)-5-甲基吡咯烷-3-醇 1108234-24-7 详细
tert-butyl (2R,4S)-4-hydroxy-2-methylpyrrolidine-1-carboxylate (2R, 4S)-4-羟基-2-甲基-吡咯烷-1-甲酸叔丁酯 348165-62-8 详细
tert-butyl (2S,4S)-4-hydroxy-2-methylpyrrolidine-1-carboxylate (2S, 4S)-4-羟基-2-甲基-吡咯烷-1-甲酸叔丁酯 477293-60-0 详细
(2S,4S)-1-(((9H-fluoren-9-yl)methoxy)carbonyl)-4-fluoropyrrolidine-2-carboxylic acid (2S,4S)-FMOC-4-氟吡咯烷-2-甲酸 203866-19-7 详细
(2S,4R)-4-fluoropyrrolidine-2-carbonitrile 1584652-40-3 详细
3-(tert-butyl) 4-methyl (S)-1,2,3-oxathiazolidine-3,4-dicarboxylate 2,2-dioxide 3-(叔丁基)4-甲基(S)-1,2,3-噁噻唑烷-3,4-二羧酸2,2-二氧化物 913979-52-9 详细
tert-butyl (2S,4S)-2-(((tert-butyldimethylsilyl)oxy)methyl)-4-hydroxypyrrolidine-1-carboxylate (3S,5S)-5-[[(叔丁基二甲基硅基)氧基]甲基]-1-BOC-吡咯烷-3-醇 216062-15-6 详细
methyl (2R,4S)-4-fluoropyrrolidine-2-carboxylate (2R,4S)-4-氟-D-脯氨酸甲酯 732957-04-9 详细
(2R,4R)-4-fluoro-2-(fluoromethyl)pyrrolidine 详细
tert-butyl (2S,4S)-2-(fluoromethyl)-4-hydroxypyrrolidine-1-carboxylate (2S,4S)-2-(氟甲基)-4-羟基吡咯烷-1-甲酸叔丁酯 1207853-00-6 详细
(2S,4S)-4-fluoropyrrolidine-2-carbonitrile hydrochloride (2S,4S)-4-氟吡咯烷-2-甲腈盐酸盐 426844-77-1 详细
(2R,4R)-1-(tert-butoxycarbonyl)-4-fluoropyrrolidine-2-carboxylic acid N-BOC-顺式-4-氟-D-脯氨酸 681128-51-8 详细
tert-butyl (S)-4-(4-fluorophenyl)-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide 叔丁基(S)-4-(4-氟苯基)-1,2,3-氧杂噻唑烷-3-羧酸酯2,2-二氧代 1379546-50-5 详细
(3S,5R)-5-(hydroxymethyl)pyrrolidin-3-ol hydrochloride (3S,5R)-5-(羟甲基)吡咯烷-3-醇盐酸盐 1018987-47-7 详细
(R)-(4,4-difluoropyrrolidin-2-yl)methanol (2R)-4,4-二氟吡咯烷-2-基]甲醇 1315691-45-2 详细
tert-butyl 4-oxa-5-thia-6-azaspiro[2.4]heptane-6-carboxylate 5,5-dioxide tert-butyl 5,5-dioxo-4-oxa-5λ-thia-6-azaspiro[2.4]heptane-6-carboxylate 2089649-97-6 详细
(2R,4S)-1-((benzyloxy)carbonyl)-4-fluoropyrrolidine-2-carboxylic acid N-CBZ-反式-4-氟-D-脯氨酸 1932069-39-0 详细
tert-butyl 4,4-dimethyl-1,2,3-oxathiazinane-3-carboxylate 2,2-dioxide 521267-13-0 详细
tert-butyl 6,6-dimethyl-1,2,3-oxathiazinane-3-carboxylate 2,2-dioxide 详细
tert-butyl (2R,4S)-2-(fluoromethyl)-4-hydroxypyrrolidine-1-carboxylate 详细
tert-butyl (2R,4S)-4-hydroxy-2-(hydroxymethyl)pyrrolidine-1-carboxylate (2R,4S)-4-羟基-2-(羟甲基)-1-吡咯烷羧酸叔丁酯 77450-03-4 详细
(2S,4R)-1-((benzyloxy)carbonyl)-4-fluoropyrrolidine-2-carboxylic acid Cbz-trans-4-fluoro-Pro-OH 72204-23-0 详细
tert-butyl (2R,4S)-4-((tert-butyldimethylsilyl)oxy)-2-(hydroxymethyl)pyrrolidine-1-carboxylate (2R,4S)-4-((叔丁基二甲基甲硅烷基)氧基)-2-(羟甲基)吡咯烷-1-羧酸叔丁酯 134441-72-8 详细
(R)-1-((benzyloxy)carbonyl)-4,4-difluoropyrrolidine-2-carboxylic acid (R)-1-((苄氧基)羰基)-4,4-二氟吡咯烷-2-羧酸 2136867-31-5 详细
tert-butyl (S)-4-(2-fluorophenyl)-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide 详细
(2S,4R)-4-fluoropyrrolidine-2-carboxylic acid hydrochloride 反式-4-氟-L-脯氨酸盐酸盐 60604-36-6 详细
(3S,5S)-5-methylpyrrolidin-3-ol hydrochloride 3-Pyrrolidinol, 5-Methyl-, hydrochloride, (3S,5S)- 1107658-77-4 详细
tert-butyl (R)-2-methyl-4-oxopyrrolidine-1-carboxylate (R)-2-甲基-4-氧代-1-吡咯烷羧酸叔丁酯 1027775-28-5 详细
tert-butyl (2S,4S)-2-(difluoromethyl)-4-hydroxypyrrolidine-1-carboxylate (2S,4S)-tert-butyl 2-(difluoromethyl)-4-hydroxypyrrolidine-1-carboxylate 1207852-93-4 详细
tert-butyl (2S,4S)-4-((tert-butyldimethylsilyl)oxy)-2-(hydroxymethyl)pyrrolidine-1-carboxylate tert-Butyl (2S,4S)-4-((tert-butyldimethylsilyl)oxy)-2-(hydroxymethyl)pyrrolidine-1-carboxylate 791602-93-2 详细
tert-butyl (R)-4-isobutyl-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide (R)-4-异丁基-1,2,3-氧杂噻唑烷-3-羧酸叔丁酯 2,2-二氧化物 1313705-90-6 详细
(S)-(4,4-difluoropyrrolidin-2-yl)methanol [(2S)-4,4-DIFLUOROPYRROLIDIN-2-YL]METHANOL 771473-90-6 详细
tert-butyl (2R,4S)-2-(((tert-butyldimethylsilyl)oxy)methyl)-4-hydroxypyrrolidine-1-carboxylate (2R,4S)-tert-butyl 2-(((tert-butyldimethylsilyl)oxy)methyl)-4-hydroxypyrrolidine-1-carboxylate 1056969-73-3 详细
tert-butyl (R)-4-((S)-sec-butyl)-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide 详细
(3R,5S)-5-(trifluoromethyl)pyrrolidin-3-ol 详细
(2S,4S)-4-fluoropyrrolidine-2-carbonitrile (2S,4S)-4-氟吡咯烷-2-甲腈 483366-10-5 详细
tert-butyl (2R,4R)-4-hydroxy-2-(hydroxymethyl)pyrrolidine-1-carboxylate (2R,4R)-4-羟基-2-(羟甲基)-1-吡咯烷羧酸叔丁酯 141850-54-6 详细
(R)-4,4-difluoropyrrolidine-2-carboxylic acid hydrochloride 6-苄氨基-1-己醇 1407991-25-6 详细
(2R,4R)-4-fluoropyrrolidine-2-carbonitrile hydrochloride (2R,4R)-顺式-4-氟-2-氰基吡咯烷盐酸盐 2306254-48-6 详细
(R)-N-(tert-butoxycarbonyl)serinic acid S,S-dioxide 1621706-88-4 详细
tert-butyl (S)-4-(methoxymethyl)-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide tert-butyl (4S)-4-(methoxymethyl)-2,2-dioxo-oxathiazolidine-3-carboxylate 2023006-41-7 详细
tert-butyl (2S,4S)-4-fluoropyrrolidine-2-carboxylate 1932331-49-1 详细
tert-butyl (R)-4,4-difluoropyrrolidine-2-carboxylate 2136231-08-6 详细
(2S,4R)-4-fluoro-2-(fluoromethyl)pyrrolidine 详细
(S)-(4,4-difluoropyrrolidin-2-yl)methanol hydrochloride (S)-(4,4-二氟吡咯烷-2-基)甲醇盐酸盐 623583-10-8 详细
methyl (2R,4R)-4-fluoropyrrolidine-2-carboxylate hydrochloride (2R,4R)-4-氟吡咯烷-2-羧酸甲酯盐酸盐 1445948-46-8 详细
tert-butyl (S)-4-(3-fluorophenyl)-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide 叔丁基(S)-4-(3-氟苯基)-1,2,3-氧杂噻唑烷-3-羧酸酯2,2-二氧代 1240480-33-4 详细
methyl (2R,4R)-4-fluoropyrrolidine-2-carboxylate 1064078-37-0 详细
((2R,4S)-4-fluoropyrrolidin-2-yl)methanol 1147181-35-8 详细
(2S,4R)-4-fluoropyrrolidine-2-carbonitrile hydrochloride (2S,4R)-反式-4-氟-2-氰基吡咯烷盐酸盐 2306249-26-1 详细
(S)-N-(tert-butoxycarbonyl)serinic acid S,S-dioxide 1620620-04-3 详细
(S)-4,4-difluoro-2-methylpyrrolidine 1670259-98-9 详细
tert-butyl 6-oxa-5-thia-4-azaspiro[2.4]heptane-4-carboxylate 5,5-dioxide 6-Oxa-5-thia-4-azaspiro[2.4]heptane-4-carboxylic acid, 1,1-dimethylethyl ester, 5,5-dioxide 2023006-14-4 详细
(2S,4S)-4-fluoro-2-methylpyrrolidine 2299230-82-1 详细
tert-butyl (2R,4S)-2-(difluoromethyl)-4-hydroxypyrrolidine-1-carboxylate 2325666-25-7 详细
tert-butyl (R)-4-(2-fluorophenyl)-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide 详细
(S)-4,4-difluoro-2-methylpyrrolidine hydrochloride 1917292-38-6 详细
4-benzyl 3-(tert-butyl) (S)-1,2,3-oxathiazolidine-3,4-dicarboxylate 2,2-dioxide 4-苄基3-(叔丁基)(S)-1,2,3-噁噻唑烷-3,4-二羧酸2,2-二氧化物 889459-00-1 详细
tert-butyl (2S,4R)-4-hydroxy-2-methylpyrrolidine-1-carboxylate (2S,4R)-4-羟基-2-甲基-吡咯烷-1-甲酸叔丁酯 114676-61-8 详细
((2R,4S)-4-fluoropyrrolidin-2-yl)methanol hydrochloride (2R,4S)-反式-4-氟-L-脯氨醇盐酸盐 1147110-60-8 详细
tert-butyl (2R,4R)-2-(((tert-butyldimethylsilyl)oxy)methyl)-4-hydroxypyrrolidine-1-carboxylate (2R,4R)-2-[[[(1,1-Dimethylethyl)dimethylsilyl]oxy]methyl]-4-hydroxy-1-pyrrolidinecarboxylic Acid 1,1-Dimethylethyl Ester 216062-16-7 详细
4-benzyl 3-(tert-butyl) (R)-1,2,3-oxathiazolidine-3,4-dicarboxylate 2,2-dioxide 4-苄基3-(叔丁基)(R)-1,2,3-噁噻唑烷-3,4-二羧酸2,2-二氧化物 1620620-29-2 详细
tert-butyl (2S,4R)-4-fluoropyrrolidine-2-carboxylate 1916479-73-6 详细
tert-butyl (S)-4-((S)-sec-butyl)-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide 1394239-78-1 详细
(R)-4,4-difluoro-2-methylpyrrolidine 1670259-97-8 详细
tert-butyl (S)-4-(difluoromethyl)-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide 详细
(3R,5R)-5-(trifluoromethyl)pyrrolidin-3-ol 2380476-61-7 详细
(S)-1-(((9H-fluoren-9-yl)methoxy)carbonyl)-4,4-difluoropyrrolidine-2-carboxylic acid (S)-1-(((9H-芴-9-基)甲氧基)羰基)-4,4-二氟吡咯烷-2-羧酸 203866-21-1 详细
tert-butyl (3aR,7aS)-hexahydro-3H-benzo[d][1,2,3]oxathiazole-3-carboxylate 2,2-dioxide (R,S)-六氢-3H-1,2,3-苯并氧杂噻唑烷-2,2-二氧-3-羧酸叔丁基酯 1206227-47-5 详细
(2S,4R)-1-(((9H-fluoren-9-yl)methoxy)carbonyl)-4-fluoropyrrolidine-2-carboxylic acid (2S,4R)-4-氟-1-FMOC-吡咯烷-2-甲酸 203866-20-0 详细
(2R,4S)-4-fluoropyrrolidine-2-carboxylic acid hydrochloride (2R,4S)-反式-4-氟-L-脯氨酸盐酸盐 1143504-73-7 详细
methyl (R)-4,4-difluoropyrrolidine-2-carboxylate (2R)-4,4-二氟吡咯烷-2-羧酸甲酯 1400688-76-7 详细
(2R,4S)-4-fluoropyrrolidine-2-carbonitrile hydrochloride (2R,4S)-反式-4-氟-2-氰基吡咯烷盐酸盐 2306247-90-3 详细
3-(tert-butyl) 4-methyl (R)-1,2,3-oxathiazolidine-3,4-dicarboxylate 2,2-dioxide (R)-3-BOC-1,2,3-氧杂噻唑烷-4-甲酸甲酯-2,2-二氧化物 1621706-89-5 详细
(3S,5R)-5-(hydroxymethyl)pyrrolidin-3-ol (3S,5R)-5-(羟甲基)吡咯烷-3-醇 825644-11-9 详细
(2R,4S)-4-fluoropyrrolidine-2-carboxylic acid (2R,4S)-4-氟吡咯烷-2-羧酸 131176-02-8 详细
tert-butyl (2R,4R)-4-fluoropyrrolidine-2-carboxylate (2R,4R)-4-氟吡咯烷-2-羧酸叔丁酯 2031242-75-6 详细
(R)-4,4-difluoro-2-methylpyrrolidine hydrochloride (R)-4,4-二氟-2-甲基吡咯烷盐酸盐 2845095-62-5 详细
(2S,4R)-4-fluoro-2-(fluoromethyl)pyrrolidine hydrochloride 详细
(2S,4R)-4-fluoropyrrolidine-2-carboxylic acid 反式-4-氟脯氨酸 2507-61-1 详细
tert-butyl (2S,4S)-4-hydroxy-2-(hydroxymethyl)pyrrolidine-1-carboxylate (2S,4S)-4-羟基-2-(羟甲基)吡咯烷-1-羧酸叔丁酯 191280-88-3 详细
tert-butyl (S)-2-methyl-4-oxopyrrolidine-1-carboxylate (S)-2-甲基-4-氧代-1-吡咯烷羧酸叔丁酯 1374673-93-4 详细
(2R,4R)-4-fluoropyrrolidine-2-carboxylic acid hydrochloride (2R,4R)-4-氟吡咯烷-2-甲酸盐酸盐 1523541-82-3 详细
(2R,4R)-4-fluoropyrrolidine-2-carboxylic acid (4R)-4-氟-D-脯氨酸 913820-71-0 详细
tert-butyl (S)-4-isobutyl-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide (S)-叔丁基 4-异丁基-1,2,3- 噁噻唑烷 -3-羧酸盐 2,2-二氧化物 1013941-87-1 详细
(2R,4S)-4-fluoropyrrolidine-2-carbonitrile 1932102-08-3 详细
(2R,4R)-4-fluoropyrrolidine-2-carbonitrile 1637365-35-5 详细
(2R,4R)-1-((benzyloxy)carbonyl)-4-fluoropyrrolidine-2-carboxylic acid N-CBZ-顺式-4-氟-D-脯氨酸 2089246-03-5 详细
tert-butyl (3aS,7aR)-hexahydro-3H-benzo[d][1,2,3]oxathiazole-3-carboxylate 2,2-dioxide 2380860-90-0 详细
(R)-5-methylpyrrolidin-3-one hydrochloride (S)-5-甲基吡咯烷-3-酮盐酸盐 2708342-87-2 详细
tert-butyl (R)-4-(3-fluorophenyl)-1,2,3-oxathiazolidine-3-carboxylate 2,2-dioxide 详细
(S)-5-methylpyrrolidin-3-one hydrochloride (R)-5-甲基吡咯烷-3-酮盐酸盐 2708343-91-1 详细
(S)-4,4-difluoropyrrolidine-2-carboxylic acid hydrochloride (S)-4,4-二氟吡咯烷-2-甲酸盐酸盐 1588480-37-8 详细
(R)-1-(((9H-fluoren-9-yl)methoxy)carbonyl)-4,4-difluoropyrrolidine-2-carboxylic acid (R)-1-(((9H-芴-9-基)甲氧基)羰基)-4,4-二氟吡咯烷-2-羧酸 273222-07-4 详细
(2R,4R)-1-(((9H-fluoren-9-yl)methoxy)carbonyl)-4-fluoropyrrolidine-2-carboxylic acid N-FMOC-顺式-4-氟-D-脯氨酸 1932387-77-3 详细
tert-butyl (2S,4R)-2-(((tert-butyldimethylsilyl)oxy)methyl)-4-hydroxypyrrolidine-1-carboxylate (2S,4R)-tert-butyl 2-(((tert-butyldimethylsilyl)oxy)methyl)-4-hydroxypyrrolidine-1-carboxylate 125653-58-9 详细
tert-butyl (S)-4,4-difluoropyrrolidine-2-carboxylate 1353053-69-6 详细
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