| Identification | Back Directory | [Name]
3-Piperidinecarboxylic acid, 1-[[4-[(diethylamino)sulfonyl]phenyl]sulfonyl]-, ethyl ester, (3R)- | [CAS]
2749554-00-3 | [Synonyms]
DX2-201
3-Piperidinecarboxylic acid, 1-[[4-[(diethylamino)sulfonyl]phenyl]sulfonyl]-, ethyl ester, (3R)- | [Molecular Formula]
C18H28N2O6S2 | [MOL File]
2749554-00-3.mol | [Molecular Weight]
432.55 |
| Hazard Information | Back Directory | [Uses]
DX2-201 is a potent and selective oxidative phosphorylation (OXPHOS) complex I inhibitor with an IC50 of 312 nM. DX2-201 has anticancer effects[1]. | [References]
[1] Ding Xue, et al. Discovery and Lead Optimization of Benzene-1,4-disulfonamides as Oxidative Phosphorylation Inhibitors.J Med Chem. 2022 Jan 13;65(1):343-368. https://pubmed.ncbi.nlm.nih.gov/34982568/ |
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