DELTORPHIN I
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- CAS号:
- 122752-15-2
- 英文名:
- DELTORPHIN I
- 英文别名:
- Delt-i;DELTORPHIN 1;DELTORPHIN C;DELTORPHIN I;Deltorphin Ⅰ;ala(2)-deltorphin;Deltorphin I(TFA);[D-ALA2]DELTORPHIN I;deltorphin I, Ala(2)-;M.W. 768.87 C37H52N8O10
- 中文名:
- DELTORPHIN I
- 中文别名:
- 化合物DELTORPHIN I(TFA);D-ALA2] DELTORPHIN I-新皮啡肽
- CBNumber:
- CB9669770
- 分子式:
- C37H52N8O10
- 分子量:
- 768.86
- MOL File:
- 122752-15-2.mol
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DELTORPHIN I化学性质
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沸点:
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1242.4±65.0 °C(Predicted)
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密度:
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1.284±0.06 g/cm3(Predicted)
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储存条件:
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-15°C
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溶解度:
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Soluble to 0.40 mg/ml in 50% acetonitrile / water
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酸度系数(pKa):
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4.19±0.10(Predicted)
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形态:
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Powder
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DELTORPHIN I性质、用途与生产工艺
Deltorphin I 是一种高亲和力的选择性 δ-阿片受体 (δ-opioid receptor) 激动剂。
Twice daily administration of Deltorphin I (20μg/mouse) for 4 days produces tolerance to Deltorphin I analgesia, as shown by the decrease in the analgesic response. The peak analgesic response to Deltorphin I (20 μg/mouse) at 10 min after injections is decreased from 8.36±0.28 s (the 1st day) to 4.53±0.14 s (the 4th day) markedly. Concurrent treatment of Melatonin (0.5, 1 and 2.5 mg/kg) and Deltorphin I (20 μg/mouse) twice daily for 4 days can attenuate the tolerance to Deltorphin I analgesia (P<0.05, <0.05 and <0.05), and this effect is dose dependent.
DELTORPHIN I
上下游产品信息
上游原料
下游产品
| 更新日期 | 产品编号 | 产品名称 | CAS编号 | 包装 | 价格 |
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| 2024/01/25 | HY-P1336 | DELTORPHIN I
Deltorphin I | 122752-15-2 | 1 mg | 800元 |
| 2024/01/25 | HY-P1336 | DELTORPHIN I
Deltorphin I | 122752-15-2 | 5 mg | 2000元 |
122752-15-2, DELTORPHIN I 相关搜索:
- Opioid receptor and opioid-like receptor
- Peptide
- 药靶配体
- 标准品
- C37H52N8O10
- D-ALA2] DELTORPHIN I-新皮啡肽
- 化合物DELTORPHIN I(TFA)
- 122752-15-2
- Glycinamide, L-tyrosyl-D-alanyl-L-phenylalanyl-L-α-aspartyl-L-valyl-L-valyl-
- Deltorphin I H-Tyr-D-Ala-Phe-Asp-Val-Val-Gly-NH2
- Deltorphin Ⅰ
- Deltorphin I(TFA)
- (3S)-3-[[(2S)-2-[[(2R)-2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]amino]-4-[[(2S)-1-[[(2S)-1-[(2-amino-2-oxoethyl)amino]-3-methyl-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-4-oxobutanoic acid
- ala(2)-deltorphin
- TYR-D-ALA-PHE-ASP-VAL-VAL-GLY-NH2
- H-TYR-D-ALA-PHE-ASP-VAL-VAL-GLY-NH2
- [D-ALA2]DELTORPHIN I
- DELTORPHIN 1
- DELTORPHIN C
- DELTORPHIN I
- deltorphin I, Ala(2)-
- Tyr-Ala-Phe-Asp-Val-val-Gly-nh2
- Glycinamide, L-tyrosyl-D-alanyl-L-phenylalanyl-L-alpha-aspartyl-L-valyl-L-valyl-
- Delt-i
- L-Tyr-D-Ala-L-Phe-L-αAsp-L-Val-L-Val-Gly-NH2
- L-Tyr-D-Ala-L-Phe-L-Asp-L-Val-L-Val-Gly-NH2
- M.W. 768.87 C37H52N8O10
- tyr-D-ala-phe-asp-val-val-gly amide