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ABCG2-IN-1

ABCG2-IN-1 structure

CAS No.: 2559759-40-7

Chemical Name:: ABCG2-IN-1

Synonyms: ABCG2-IN-1;Pyrazino[1′,2′:1,6]pyrido[3,4-b]indole-3-propanamide, N-(1,1-dimethylethyl)-1,2,3,4,6,7,12,12a-octahydro-9-methoxy-6-(2-methylpropyl)-1,4-dioxo-, (3S,6S,12aS)-

CBNumber:: CB014133772

Molecular Formula:: C26H36N4O4

Molecular Weight:: 468.59

MDL Number:

MOL File:: 2559759-40-7.mol

Last updated:2025-05-19 13:47:39

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ABCG2-IN-1 Properties

Boiling point	767.425±60.00 °C(Press: 760.00 Torr)(predicted)
Density	1.236±0.10 g/cm3(Temp: 25 °C; Press: 760 Torr)(predicted)
pka	13.360±0.60(predicted)

ABCG2-IN-1 Chemical Properties,Uses,Production

Uses

ABCG2-IN-1 (compound K2), a Ko143 analog, is an orally active ABCG2 inhibitor with an IC50 of 0.13 μM. ABCG2-IN-1 has favorable oral pharmacokinetic profiles in mice[1].

References

[1] Junjie Zhu, et al. Metabolism-guided development of Ko143 analogs as ABCG2 inhibitors. Eur J Med Chem. 2023 Nov 5;259:115666. DOI:10.1016/j.ejmech.2023.115666

ABCG2-IN-1 Preparation Products And Raw materials

Raw materials

Preparation Products

ABCG2-IN-1 Suppliers

Global( 2)Suppliers

Supplier	Tel	Email	Country	ProdList	Advantage
TargetMol Chemicals Inc.	+17819995354	marketing@targetmol.com	United States	19939	58
TargetMol Chemicals Inc.	15002134094	marketing@targetmol.cn	China	26070	58

Supplier	Advantage
TargetMol Chemicals Inc.	58
TargetMol Chemicals Inc.	58

View Lastest Price from ABCG2-IN-1 manufacturers

Image	Update time	Product	Price	Min. Order	Purity	Supply Ability	Manufacturer
	2025-04-29	ABCG2-IN-1 2559759-40-7	US $1980.00-1520.00 / mg			10g	TargetMol Chemicals Inc.

ABCG2-IN-1
2559759-40-7
US $1980.00-1520.00 / mg
TargetMol Chemicals Inc.

ABCG2-IN-1 Pyrazino[1′,2′:1,6]pyrido[3,4-b]indole-3-propanamide, N-(1,1-dimethylethyl)-1,2,3,4,6,7,12,12a-octahydro-9-methoxy-6-(2-methylpropyl)-1,4-dioxo-, (3S,6S,12aS)- 2559759-40-7