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CAPSAZEPINE

CAPSAZEPINE
CAPSAZEPINE
CAS No.
138977-28-3
Chemical Name:
CAPSAZEPINE
Synonyms
CAPSAZEPINE;Capsazepine,98%;CAPSAZEPINE SYNTHETIC ANALOG OF C;2-[[2-(4-Chlorophenyl)ethylamino]thiocarbonyl]-2,3,4,5-tetrahydro-1H-2-benzazepine-7,8-diol;N-[2-(CHLOROPHENYL)ETHYL]-1,3,4,5-TETRAHYDRO-7,8-DIHYDROXY-2H-2-BENZAZEPINE-2-CARBOTHIOAMIDE;N-[2-(4-CHLOROPHENYL)ETHYL]-1,3,4,5-TETRAHYDRO-7,8-DIHYDROXY-2H-2-BENZAZEPINE-2-CARBOTHIOAMIDE
CBNumber:
CB0144302
Molecular Formula:
C19H21ClN2O2S
Formula Weight:
376.9
MOL File:
138977-28-3.mol

CAPSAZEPINE Properties

Melting point:
155-157°C
storage temp. 
2-8°C
solubility 
methanol: soluble
form 
solid
color 
off-white
InChIKey
DRCMAZOSEIMCHM-UHFFFAOYSA-N
CAS DataBase Reference
138977-28-3(CAS DataBase Reference)

SAFETY

Hazard Codes  Xn
Risk Statements  20/21/22-36/37/38
Safety Statements  22-24/25-36-26
RIDADR  2811
WGK Germany  3
HazardClass  6.1(a)
PackingGroup  II

CAPSAZEPINE price More Price(8)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Sigma-Aldrich C191 Capsazepine ≥98% (HPLC), solid 138977-28-3 5mg $186 2018-11-13 Buy
Sigma-Aldrich C191 Capsazepine ≥98% (HPLC), solid 138977-28-3 25mg $657 2018-11-13 Buy
Alfa Aesar J63055 Capsazepine, 99+% 138977-28-3 50mg $1284 2018-11-13 Buy
Alfa Aesar J63055 Capsazepine, 99+% 138977-28-3 10mg $300 2018-11-13 Buy
Cayman Chemical 10007518 Capsazepine ≥98% 138977-28-3 1mg $25 2018-11-19 Buy

CAPSAZEPINE Chemical Properties,Uses,Production

Chemical Properties

Light Yellow Solid

Uses

A selective vanilloid receptor antagonist (Ki=3.2uM

Definition

ChEBI: A benzazepine that is 2,3,4,5-tetrahydro-1H-2-benzazepine which is substituted by hydroxy groups at positions 7 and 8 and on the nitrogen atom by a 2-(p-chlorophenyl)ethylaminothiocarbonyl group. A synthetic analogue of caps icin, it was the first reported capsaicin receptor antagonist.

Hazard

A poison.

Biological Activity

Selective vanilloid receptor antagonist (K i = 3.2 μ M). Inhibits carrageenan inflammation-induced hyperalgesic responses in the rat. Also activates amiloride-sensitive epithelial Na + channel ENaC δ . Also available as part of the Vanilloid TRPV1 Receptor Tocriset™ .

CAPSAZEPINE Preparation Products And Raw materials

Raw materials

Preparation Products


CAPSAZEPINE Suppliers

Global( 73)Suppliers
Supplier Tel Fax Email Country ProdList Advantage
Mainchem Co., Ltd.
+86-0592-6210733
+86-0592-6210733 sales@mainchem.com CHINA 32651 55
ATK CHEMICAL COMPANY LIMITED
+86 21 5161 9050/ 5187 7795
+86 21 5161 9052/ 5187 7796 ivan@atkchemical.com CHINA 14293 60
Ningbo Materials-X Co., Ltd 0574-87487840-805 15888368997
0574-87485342 sales@mater-x.com China 475 55
J & K SCIENTIFIC LTD. 400-666-7788 +86-10-82848833
+86-10-82849933 jkinfo@jkchemical.com;market6@jkchemical.com China 96815 76
3B Pharmachem (Wuhan) International Co.,Ltd. 86-21-50328103 * 801、802、803、804 Mobile:18930552037
86-21-50328109 3bsc@sina.com China 15926 69
Ascent Scientific 4401179829988
4402030 700 369 customerservice@ascentscientific.co.uk United Kingdom 280 60
Nanjing Chemlin Chemical Co., Ltd 025-83697070
+86-25-83453306 sales@chemlin.com.cn China 19998 64
Chemsky(shanghai)International Co.,Ltd. 021-50135380
shchemsky@sina.com China 32492 50
Jinan Haohua Industry Co., Ltd 0531-58773082 ;58773060
0531-58773099 sales@jnhaohua.com China 5621 58
Shanghai LiuShi Pharmaceutical Technology Co., Ltd. 021-60135539
021-38721356 shlschemical@hotmail.com China 9947 55

138977-28-3(CAPSAZEPINE)Related Search:


  • CAPSAZEPINE
  • N-[2-(CHLOROPHENYL)ETHYL]-1,3,4,5-TETRAHYDRO-7,8-DIHYDROXY-2H-2-BENZAZEPINE-2-CARBOTHIOAMIDE
  • N-[2-(4-CHLOROPHENYL)ETHYL]-1,3,4,5-TETRAHYDRO-7,8-DIHYDROXY-2H-2-BENZAZEPINE-2-CARBOTHIOAMIDE
  • CAPSAZEPINE SYNTHETIC ANALOG OF C
  • 2-[[2-(4-Chlorophenyl)ethylamino]thiocarbonyl]-2,3,4,5-tetrahydro-1H-2-benzazepine-7,8-diol
  • Capsazepine,98%
  • 138977-28-3
  • C19H21ClN2O2S
  • Inhibitors
  • Intermediates & Fine Chemicals
  • Pharmaceuticals
  • Vanilloid/TRPV channel
  • Ion Channels
  • Amines
  • Aromatics
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