ChemicalBook >> CAS DataBase List >>GSK962040
GSK962040
- CAS No.
- 923565-21-3
- Chemical Name:
- GSK962040
- Synonyms
- Camicil;Camicinal;GSK962040;Lopixibat chloride;GSK962040 (Camicinal;1-[4-[(3-Fluorophenyl)amino]-1-piperidinyl]-2-[4-[[(3S)-3-methyl-1-piperazinyl]methyl]phenyl]ethanone;Ethanone, 1-[4-[(3-fluorophenyl)amino]-1-piperidinyl]-2-[4-[[(3S)-3-methyl-1-piperazinyl]methyl]phenyl]-
- CBNumber:
- CB02627933
- Molecular Formula:
- C25H33FN4O
- Molecular Weight:
- 424.55
- MDL Number:
- MOL File:
- 923565-21-3.mol
- MSDS File:
- SDS
Last updated:2023-05-21 10:59:17
| Melting point | 144℃ |
|---|---|
| Boiling point | 610.0±55.0 °C(Predicted) |
| Density | 1.175±0.06 g/cm3(Predicted) |
| storage temp. | Store at -20°C |
| solubility | Soluble in DMSO |
| pka | 9.21±0.40(Predicted) |
| FDA UNII | 3C8348951H |
SAFETY
Risk and Safety Statements
| Symbol(GHS) |  GHS07 |
|---|---|
| Signal word | Warning |
| Hazard statements | H302 |
| Precautionary statements | P264-P270-P301+P312-P330-P501 |
GSK962040 price
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| ChemScene | CS-2312 | Camicinal 95.82% | 923565-21-3 | 10mg | $600 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0013933 | GSK-962040 95.00% | 923565-21-3 | 5MG | $660 | 2021-12-16 | Buy |
| ChemScene | CS-2312 | Camicinal 95.82% | 923565-21-3 | 5mg | $420 | 2021-12-16 | Buy |
| ApexBio Technology | B1149 | GSK962040 | 923565-21-3 | 5mg | $512 | 2021-12-16 | Buy |
| ChemScene | CS-2312 | Camicinal 95.82% | 923565-21-3 | 50mg | $1800 | 2021-12-16 | Buy |
GSK962040 Chemical Properties,Uses,Production
Definition
ChEBI: Camicinal is a member of acetamides.
Biological Activity
Camicinal (GSK962040) is a motilin receptor agonist with a pEC50 of 7.9.
in vivo
Camicinal (GSK962040) (5 mg free base kg 1) also produced an increase in total faecal weight over the 2-h postdose period (21.2 ± 4.5 g; P < 0.05). It induced phasic contractions, the duration of which was dose-related (48 and 173 min for 3 and 6 mg kg 1), driven by mean plasma concentrations >1.14 μmol L 1. After the effects of GSK962040 faded, migrating motor complex (MMC) activity returned.
target
pEC50: 7.9 (Motilin Receptor).
GSK962040 Preparation Products And Raw materials
Raw materials
Preparation Products
GSK962040 Suppliers
Global( 32)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| TargetMol Chemicals Inc. | +1-781-999-5354 +1-00000000000 | marketing@targetmol.com | United States | 19892 | 58 |
| Career Henan Chemica Co | +86-0371-86658258 15093356674; | laboratory@coreychem.com | China | 30255 | 58 |
| InvivoChem | +1-708-310-1919 +1-13798911105 | sales@invivochem.cn | United States | 6393 | 58 |
| Amadis Chemical Company Limited | 571-89925085 | sales@amadischem.com | China | 131981 | 58 |
| Haoyuan Chemexpress Co., Ltd. | 021-58950125 | info@chemexpress.com | China | 7553 | 61 |
| LETOPHARM LIMITED | +86-21-5821 5861 | sales@letopharm.com | China | 2384 | 58 |
| SPIRO PHARMA | eric_feng1954@126.com | China | 9254 | 55 | |
| Guangzhou QiYun Biotechnology Co., Ltd. | 020-61288194 61288195 | 505721671@qq.com | China | 3868 | 58 |
| Musechem | +1-800-259-7612 | info@musechem.com | United States | 4662 | 60 |
| Fan De(Beijing) Biotechnology Co., Ltd. | 15911056312 | liming@bio-fount.com | China | 9730 | 58 |
| Supplier | Advantage |
|---|---|
| TargetMol Chemicals Inc. | 58 |
| Career Henan Chemica Co | 58 |
| InvivoChem | 58 |
| Amadis Chemical Company Limited | 58 |
| Haoyuan Chemexpress Co., Ltd. | 61 |
| LETOPHARM LIMITED | 58 |
| SPIRO PHARMA | 55 |
| Guangzhou QiYun Biotechnology Co., Ltd. | 58 |
| Musechem | 60 |
| Fan De(Beijing) Biotechnology Co., Ltd. | 58 |
GSK962040
1-[4-[(3-Fluorophenyl)amino]-1-piperidinyl]-2-[4-[[(3S)-3-methyl-1-piperazinyl]methyl]phenyl]ethanone
Camicinal
Lopixibat chloride
GSK962040
(Camicinal
Camicil
Ethanone, 1-[4-[(3-fluorophenyl)amino]-1-piperidinyl]-2-[4-[[(3S)-3-methyl-1-piperazinyl]methyl]phenyl]-
923565-21-3
C25H33FN4O