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GF109203X

GF109203X
GF109203X structure
CAS No.
133052-90-1
Chemical Name:
GF109203X
Synonyms
BIM 1;GO 6850;G 6850];GF 109203X;GO 6850 HCL;GF-109203X HCL;BISINDOYLMALEIMIDE;BISINDOLYLMALEIMIDE;BISINDOLYLMALEIMIDE I;Bisindolylmaleinimide
CBNumber:
CB2103079
Molecular Formula:
C25H24N4O2
Formula Weight:
412.48
MOL File:
133052-90-1.mol

GF109203X Properties

Melting point:
280℃ (decomposition)
storage temp. 
2-8°C
solubility 
DMSO: ~1 mg/mlsoluble
form 
Liquid
Water Solubility 
Insoluble in water.
SAFETY
  • Risk and Safety Statements
  • Hazard and Precautionary Statements (GHS)
Hazard Codes  Xn
Risk Statements  40-22
Safety Statements  36/37
WGK Germany  3
RTECS  UX9590000
Symbol(GHS):
Signal word: Warning
Hazard statements:
Code Hazard statements Hazard class Category Signal word Pictogram P-Codes
H351 Suspected of causing cancer Carcinogenicity Category 2 Warning P201, P202, P281, P308+P313, P405,P501
Precautionary statements:
P280 Wear protective gloves/protective clothing/eye protection/face protection.

GF109203X price More Price(9)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Sigma-Aldrich 203290 Bisindolylmaleimide I 133052-90-1 250ug $53.6 2018-11-20 Buy
Sigma-Aldrich 203290 Bisindolylmaleimide I 133052-90-1 1mg $141 2018-11-20 Buy
Alfa Aesar J63401 Bisindolylmaleimide 1 133052-90-1 25mg $427 2018-11-13 Buy
Alfa Aesar J63401 Bisindolylmaleimide 1 133052-90-1 5mg $120 2018-11-13 Buy
Cayman Chemical 13298 Bisindolylmaleimide I ≥95% 133052-90-1 10mg $131 2018-11-13 Buy

GF109203X Chemical Properties,Uses,Production

Biological Activity

Very potent and selective inhibitor of protein kinase C, selective for the α and β 1 isoforms (IC 50 values are 0.0084, 0.0180, 0.210, 0.132, and 5.8 μ M for α , β 1, δ , ε , and ζ isoforms respectively). Selective over MLCK, PKG and PKA (IC 50 values are 0.6, 4.6, and 33 μ M respectively). Potent antagonist at the 5-HT 3 receptor (K i = 29.5 nM). Anti-inflammatory in vivo . Also available as part of the Mixed Kinase Inhibitor Tocriset™ .

GF109203X Preparation Products And Raw materials

Raw materials

Preparation Products


GF109203X Suppliers

Global( 74)Suppliers
Supplier Tel Fax Email Country ProdList Advantage
ATK CHEMICAL COMPANY LIMITED
+86 21 5161 9050/ 5187 7795
+86 21 5161 9052/ 5187 7796 ivan@atkchemical.com CHINA 16534 60
Biochempartner
0086-13720134139
candy@biochempartner.com CHINA 956 58
J & K SCIENTIFIC LTD. 400-666-7788 +86-10-82848833
+86-10-82849933 jkinfo@jkchemical.com;market6@jkchemical.com China 96815 76
3B Pharmachem (Wuhan) International Co.,Ltd. 86-21-50328103 * 801、802、803、804 Mobile:18930552037
86-21-50328109 3bsc@sina.com China 15926 69
VDM Biochemicals 0330-2528181
0330-2528171 sales@vdmbio.com United States 511 64
Jinan Trio PharmaTech Co., Ltd. +86 (531) 88811783;
+86 (531) 55696010 QQ 1762738062 sales@trio-pharmatech.com (International market);trio@trio-pharmatech.com(Domestic market) China 1858 62
Sinopharm Chemical Reagent Co,Ltd. 86-21-63210123
86-21-63290778 86-21-63218885 sj_scrc@sinopharm.com China 9966 79
SpringPharma Tech Co.,Ltd +86-25-68710855/ +86-25-68710897
025-68710856 sales@springpharma.net China 1264 62
BOC Sciences
info@bocsci.com United States 10558 65
Shanghai LiuShi Pharmaceutical Technology Co., Ltd. 021-60135539
021-38721356 shlschemical@hotmail.com China 9947 55

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