GR 89696 FUMARATE
- CAS No.
- 126766-32-3
- Chemical Name:
- GR 89696 FUMARATE
- Synonyms
- GR 89696;GR 89696 FUMARATE;GR 89696 fumarate salt solid;GR 89696 fumarate, 10 mM in DMSO;Methyl 4-(2-(3,4-dichlorophenyl)acetyl)-3-(pyrrolidin-1-ylmethyl)piperazine-1-carboxylate fumarate;4-((3,4-Dichlorophenyl)acetyl)-3-(1-pyrrolidinylmethyl)-1-piperazinecarboxylicacidmethylesterfumarate;4-([3,4-DICHLOROPHENYL]ACETYL)-3-(1-PYRROLIDINYLMETHYL)-1-PIPERAZINECARBOXYLIC ACID METHYL ESTER FUMARATE
- CBNumber:
- CB4178514
- Molecular Formula:
- C23H29Cl2N3O7
- Molecular Weight:
- 530.4
- MDL Number:
- MOL File:
- 126766-32-3.mol
| storage temp. | Store at RT |
|---|---|
| solubility | ethanol: 4.0 mg/mL |
| form | solid |
| color | off-white |
| FDA UNII | YDF52K5SDR |
| UNSPSC Code | 12352200 |
| NACRES | NA.77 |
GR 89696 FUMARATE price More Price(9)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Sigma-Aldrich | G133 | GR 89696 fumarate salt solid | 126766-32-3 | 25mg | $490 | 2025-07-31 | Buy |
| Tocris | 1483 | GR89696fumarate ≥99%(HPLC) | 126766-32-3 | 10 | $175 | 2021-12-16 | Buy |
| Tocris | 1483 | GR89696fumarate ≥99%(HPLC) | 126766-32-3 | 50 | $737 | 2021-12-16 | Buy |
| Usbiological | 255397 | GR 89696 fumarate | 126766-32-3 | 10mg | $423 | 2021-12-16 | Buy |
| TRC | G779535 | GR89696 | 126766-32-3 | 5mg | $1425 | 2021-12-16 | Buy |
GR 89696 FUMARATE Chemical Properties,Uses,Production
Uses
GR 89696 is a selective κ-opioid receptor agonist with anti-nociceptive and neuroprotective properties.
Biological Activity
Highly potent and selective κ -opioid agonist (IC 50 = 0.04 nM) that may be selective for the putative κ 2 receptor. Anti-nociceptive and neuroprotective in vivo .
in vivo
GR 89696 (intramuscular injection, 0.01-0.1 μg/kg) attenuates the scratching response induced by intrathecal morphine (0.03mg) in a dose-dependent manner without affecting the analgesic effect of morphine[1].
GR-896960(subcutaneous injection, 1 mg/kg) reduces cerebral artery infarct volume by 38% in a rat model of permanent focal ischemia[2].
storage
Store at +4°C
GR 89696 FUMARATE Preparation Products And Raw materials
Raw materials
Preparation Products
GR 89696 FUMARATE Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| TargetMol Chemicals Inc. | +1-781-999-5354; +17819995354 | marketing@targetmol.com | United States | 32376 | 58 |
| Aladdin Scientific | tp@aladdinsci.com | United States | 57505 | 58 | |
| Wuhan Jingkang en Biomedical Technology Co., Ltd | +8613720134139 | orders@jknbiochem.com | China | 5221 | 58 |
| DAYANG CHEM (HANGZHOU) CO.,LTD | +86-88938639 +86-17705817739 | info@dycnchem.com | China | 53900 | 58 |
| 3B Pharmachem (Wuhan) International Co.,Ltd. | 821-50328103-801 18930552037 | 3bsc@sina.com | China | 15839 | 69 |
| Shanghai Lollane Biological Technology Co.,Ltd. | 021-52996696，15000506266 15000506266 | China | 4649 | 55 | |
| EMMX Biotechnology LLC | 888-539-0666 | info@emmx.com | United States | 8447 | 60 |
| Shanghai EFE Biological Technology Co., Ltd. | 021-65675885 18964387627 | info@efebio.com | China | 9803 | 58 |
| Shanghai YuanYe Biotechnology Co., Ltd. | 021-61312847; 18021002903 | 3008007409@qq.com | China | 71826 | 60 |
| Shanghai Chaolan Chemical Technology Center | 021-QQ：65489617 15618227136 | Sales@ATKchemical.com | China | 9364 | 58 |
View Lastest Price from GR 89696 FUMARATE manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
 |
2025-04-30 | GR 89696 fumarate
126766-32-3
|
US $58.00-165.00 / mg | 99.19% | 10g | TargetMol Chemicals Inc. |
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- GR 89696 fumarate
126766-32-3
- US $58.00-165.00 / mg
- 99.19%
- TargetMol Chemicals Inc.