ChemicalBook >> CAS DataBase List >>RJR-2429 2HCL
RJR-2429 2HCL
- CAS No.
- 91556-75-1
- Chemical Name:
- RJR-2429 2HCL
- Synonyms
- RJR-2429 2HCL;1-Azabicyclo[2.2.2]octane, 2-(3-pyridinyl)-
- CBNumber:
- CB4497095
- Molecular Formula:
- C12H16N2
- Molecular Weight:
- 188.27
- MDL Number:
- MOL File:
- 91556-75-1.mol
Last updated:2023-04-23 13:52:06
| Boiling point | 295.6±15.0 °C(Predicted) |
|---|---|
| Density | 1.11±0.1 g/cm3(Predicted) |
| storage temp. | Desiccate at RT |
| solubility | H2O: 5 mg/mL |
| pka | 9.41±0.40(Predicted) |
| form | solid |
| color | white |
| FDA UNII | Q2L6T24QLT |
RJR-2429 2HCL Chemical Properties,Uses,Production
Uses
RJR 2429 is a potent AChR agonist.
Biological Activity
Potent nAChR agonist that displays selectivity for α 4 β 2 (K i = 1 nM) and α 1 β γ δ subtypes (EC 50 values are 297 and 55 nM respectively). Induces dopamine release from striatal neurons (EC 50 = 2 nM) and inhibits ion flux in thalamic neurons (IC 50 = 154 nM). Also putative α 3 β 4 agonist that potentiates catecholamine release.
RJR-2429 2HCL Preparation Products And Raw materials
Raw materials
Preparation Products
RJR-2429 2HCL Suppliers
Global( 4)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| 3B Pharmachem (Wuhan) International Co.,Ltd. | 821-50328103-801 18930552037 | 3bsc@sina.com | China | 15848 | 69 |
| EMMX Biotechnology LLC | 888-539-0666 | info@emmx.com | United States | 8449 | 60 |
| Supplier | Advantage |
|---|---|
| 3B Pharmachem (Wuhan) International Co.,Ltd. | 69 |
| EMMX Biotechnology LLC | 60 |
RJR-2429 2HCL
1-Azabicyclo[2.2.2]octane, 2-(3-pyridinyl)-
91556-75-1