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RX 821002

RX 821002 structure

CAS No.: 102575-24-6

Chemical Name:: RX 821002

Synonyms: Rx 821001;RX821002HCl;2-methoxyidazoxan;RX 821002 hydrochlor;2-[2-(2-methoxy-1,4-benzodioanyl)]-imidazoline hydrochloride;2-(3-methoxy-2H-1,4-benzodioxin-3-yl)-4,5-dihydro-1H-imidazole;2-(2,3-Dihydro-2-methoxy-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole;1H-Imidazole, 2-(2,3-dihydro-2-methoxy-1,4-benzodioxin-2-yl)-4,5-dihydro-

CBNumber:: CB9498390

Molecular Formula:: C12H14N2O3

Molecular Weight:: 234.25

MDL Number:

MOL File:: 102575-24-6.mol

Last updated:2023-04-23 13:52:06

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RX 821002 Properties

Boiling point	407.9±45.0 °C(Predicted)
Density	1.34±0.1 g/cm3(Predicted)
storage temp.	Desiccate at RT
form	solid
pka	9.51±0.40(Predicted)
color	white
EWG's Food Scores	1
FDA UNII	E27LB7P0ET

SAFETY

Risk and Safety Statements

Hazard Codes	Xi
Risk Statements	36/37/38
Safety Statements	26-36
WGK Germany	3

RX 821002 Chemical Properties,Uses,Production

Definition

ChEBI: A benzodioxine that is idazoxan substituted at position 2 by a methoxy group.

Biological Activity

Potent, selective α 2 -adrenoceptor antagonist with very low affinity for imidazoline sites. Displays selectivity for the α 2D over the α 2A subtypes (pK d values are 9.7 and 8.2 respectively).

RX 821002 synthesis

Synthesis of RX 821002 from 2,3-DIHYDRO-1,4-BENZODIOXINE-2-CARBONITRILE

RX 821002 Preparation Products And Raw materials

Raw materials

1,4-Benzodioxin-2-carbonitrile, 2-bromo-2,3-dihydro- 2,3-DIHYDRO-1,4-BENZODIOXINE-2-CARBONITRILE

Preparation Products

RX 821002 Suppliers

Global( 13)Suppliers

Supplier	Tel	Email	Country	ProdList	Advantage
TargetMol Chemicals Inc.	+1-781-999-5354 +1-00000000000	marketing@targetmol.com	United States	19892	58
3B Pharmachem (Wuhan) International Co.,Ltd.	821-50328103-801 18930552037	3bsc@sina.com	China	15848	69
EMMX Biotechnology LLC	888-539-0666	info@emmx.com	United States	8449	60
Suzhou Rovathin Foreign Trade Co.,Ltd	0512-65816829 18662214788	info@rovathin.com.cn	China	9332	58
Shanghai Dexuan Pharmaceutical Technology Co., Ltd	1701086315	dexuanpharma@126.com	China	9478	58
Shanghai Universal Biotech Co.,Ltd	18768175414	gaojun@univ-bio.com	China	24998	58
TargetMol Chemicals Inc.	4008200310	marketing@tsbiochem.com	China	24131	58

Supplier	Advantage
TargetMol Chemicals Inc.	58
3B Pharmachem (Wuhan) International Co.,Ltd.	69
EMMX Biotechnology LLC	60
Suzhou Rovathin Foreign Trade Co.,Ltd	58
Shanghai Dexuan Pharmaceutical Technology Co., Ltd	58
Shanghai Universal Biotech Co.,Ltd	58
TargetMol Chemicals Inc.	58

RX821002HCl 2-[2-(2-methoxy-1,4-benzodioanyl)]-imidazoline hydrochloride 2-methoxyidazoxan 1H-Imidazole, 2-(2,3-dihydro-2-methoxy-1,4-benzodioxin-2-yl)-4,5-dihydro- 2-(2,3-Dihydro-2-methoxy-1,4-benzodioxin-2-yl)-4,5-dihydro-1H-imidazole Rx 821001 2-(3-methoxy-2H-1,4-benzodioxin-3-yl)-4,5-dihydro-1H-imidazole RX 821002 hydrochlor 102575-24-6 Adrenoceptor