FGF-401 化学特性,用途語,生産方法
説明
FGF401 is an inhibitor of FGF receptor 4 (FGFR4; IC
50 = 1.9 nM). It inhibits proliferation of Huh7 carcinoma cells with an IC
50 value of 12 nM. FGF401 induces bile acid synthesis in dogs, increasing plasma and fecal levels of bile acids when administered at a dose of 45 mg/kg per day for four weeks. It also decreases serum cholesterol when administered at doses ranging from 5 to 45 mg/kg per day.
FGF-401 上流と下流の製品情報
原材料
準備製品