2-[[[2-(Tetradecyl)phenyl]amino]carbonyl]benzoic acid 化学特性,用途語,生産方法
使用
CX08005 is a competitive PTP1B inhibitor (IC50 = 0.781 μM). Binds catalytic P-loop of enzyme. Improves insulin sensitivity in obese mice in the glucose tolerance test and the homeostasis model assessment of insulin resistance index (HOMA-IR). Enhances insulin-induced glucose uptake in adipocytes and myotubes in vitro. Exhibits some selectivity for PTP1B over other protein tyrosine phosphatases, except TCPTP.
2-[[[2-(Tetradecyl)phenyl]amino]carbonyl]benzoic acid 上流と下流の製品情報
原材料
準備製品