8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride

591771-91-4

CAS番号.: 591771-91-4

化学名:

别名:

英語名:: 8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride

英語别名:: PSB 10;PSB 10 HYDROCHLORIDE;8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride

CBNumber:: CB4842011

化学式:: C16H14Cl3N5O.ClH

分子量:: 435.141

MOL File:: 591771-91-4.mol

物理性質

安全性情報

価格2

用途語

生産企業 16

8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride 物理性質

貯蔵温度 :: Desiccate at +4°C

溶解性:: Soluble to 25 mM in DMSO and to 10 mM in ethanol

外見 :: Powder

安全性情報

HSコード	2933990099

8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride 価格もっと(2)

メーカー	製品番号	製品説明	CAS番号	包装	価格	更新時間	購入
富士フイルム和光純薬株式会社(wako)	W01TOC2010	PSB 10 hydrochloride	591771-91-4	10mg	￥74000	2024-03-01	購入
富士フイルム和光純薬株式会社(wako)	W01TOC2010	PSB 10 hydrochloride	591771-91-4	50mg	￥313000	2024-03-01	購入

8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride 化学特性,用途語,生産方法

生物活性

Potent and highly selective antagonist for the human adenosine A 3 receptor, with low affinity for the rat A 3 receptor (K i values are 0.44 and > 17000 nM respectively). Displays > 3800-fold selectivity over human A 1 , A 2A and A 2B receptors (K i values are 4.1, 3.3 and 30 μ M respectively) and > 1800-fold selectivity over rat A 1 and A 2A receptors. Acts as an inverse agonist in the [ 35 S]GTP γ S binding assay in hA 3 -CHO cells (IC 50 = 4 nM). Produces thermal hyperalgesia in mice in vivo .

8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride 上流と下流の製品情報

原材料

準備製品

8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride 生産企業

Global( 16)Suppliers

名前	電話番号	電子メール	国籍	製品カタログ	優位度
3B Pharmachem (Wuhan) International Co.,Ltd.	18930552037	3bsc@sina.com	China	15813	69
EMMX Biotechnology LLC	888-539-0666	info@emmx.com	United States	8435	60
TargetMol Chemicals Inc.	+1-781-999-5354; +1-00000000000	marketing@targetmol.com	United States	32431	58
TargetMol Chemicals Inc.	4008200310 15002144251	marketing@tsbiochem.com	China	24951	58
Shanghai Tachizaki Biomedical Research Center	18014399201	sales@chemlab-tachizaki.com	China	2934	58
Aladdin Scientific		tp@aladdinsci.com	United States	50068	58

591771-91-4()キーワード:

5'-デオキシ-5'-オキソ-5'-(エチルアミノ)アデノシン 6-(2-クロロ-6-メチル-4-ピリジル)-5-(4-フルオロフェニル)-1,2,4-トリアジン-3-アミン N,N-ジメチルアデノシン 1-プロピル-8-[4-[[4-(4-クロロフェニル)ピペラジノ]スルホニル]フェニル]キサンチン 5-アミノ-9-クロロ-2-(2-フラニル)[1,2,4]トリアゾロ[1,5-c]キナゾリン