RS39604塩酸塩 化学特性,用途語,生産方法
使用
RS 39604 Hydrochloride is a potent, selective and orally active 5-HT4 receptor antagonist.
生物活性
A potent and selective 5-HT 4 antagonist, with a pK i of 9.1 at 5-HT 4 receptors in guinea pig striatal membranes and greater than 1000-fold selectivity over 5-HT 1A, 2C, 3 and D 1 , D 2 , M 1 , M 2 , AT 1, B 1 and α 1C receptors. The ketone group gives RS 39604 a relatively long half life; it is also orally active and so suitable for in vivo studies.
RS39604塩酸塩 上流と下流の製品情報
原材料
準備製品