NF110

NF110 구조식 이미지
카스 번호:
111150-22-2
상품명:
NF110
동의어(영문):
NF110;4,4',4'',4'''-[Carbonylbis[imino-5,1,3-benzenetriylbis(carbonylimino)]]tetrakisbenzenesulfonicacidtetrasodiumsalt;4-[[3-[[3,5-bis[(4-sulfonatophenyl)carbamoyl]phenyl]carbamoylamino]-5-[(4-sulfonatophenyl)carbamoyl]benzoyl]amino]benzenesulfonate
CBNumber:
CB0838926
분자식:
C41H28N6O17S4.4Na
포뮬러 무게:
1096.92
MOL 파일:
111150-22-2.mol

NF110 속성

저장 조건
Desiccate at RT
물리적 상태
가루
수용성
Soluble to 40 mM in water

안전

NF110 C화학적 특성, 용도, 생산

용도

NF 110 is a potent P2X3 receptor antagonist.

생물학적 활성

High affinity P2X 3 receptor antagonist (K i values are 36, 82 and 4144 nM for P2X 3 , P2X 1 and P2X 2 recombinant receptors respectively). Shows no activity at P2Y 1 , P2Y 2 and P2Y 11 receptors (IC 50 > 10 μ M). Potently inhibits α , β -meATP-evoked desensitizing currents in rat DRG neurons (IC 50 = 527 nM). Shows antitumor activity against several tumor types.

NF110 준비 용품 및 원자재

원자재

준비 용품


NF110 공급 업체

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