Flupirtine maleate is a centrally-acting, non-addicting analgesic agent somewhat
more potent than aspirin, paracetamol and pentazocine. It is reported to be
useful in the treatment of postoperative and dental pain.
화학적 성질
Off-White Solid
용도
Analgesic. Substituted pyridine with central analgesic properties.
생물학적 활성
Non-opioid analgesic with muscle relaxant properties. Activates K + channels and indirectly antagonizes NMDA receptors. Exhibits neuroprotective actions in a model of cerebral ischemia in mice and reduces apoptosis and necrosis induced by noxious stimuli.
