PD 135158

PD 135158 구조식 이미지
카스 번호:
130325-35-8
상품명:
PD 135158
동의어(영문):
PD 135158;4-[[(1R)-2-[[(2R)-3-(1H-Indol-3-yl)-2-methyl-1-oxo-2-[[[[(1S,2R,4S)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]oxy]carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoicacid
CBNumber:
CB41400397
분자식:
C42H61N5O11
포뮬러 무게:
811.97
MOL 파일:
130325-35-8.mol

PD 135158 속성

저장 조건
Store at +4°C
용해도
<61.68mg/ml in DMSO

안전

PD 135158 C화학적 특성, 용도, 생산

생물학적 활성

Potent and selective, nonpeptide CCK 2 receptor antagonist (IC 50 values are 2.8 and 1232 nM for CCK 2 and CCK 1 respectively) that displays negligible affinity at GABA A , benzodiazepine, substance P, neurotensin, opioid, bradykinin and 5-HT 3 receptors (IC 50 > 10 μ M). Exhibits anxiolytic activity in elevated plus maze and social interaction tests and increases food intake in rats.

PD 135158 준비 용품 및 원자재

원자재

준비 용품


PD 135158 공급 업체

글로벌( 16)공급 업체
공급자 전화 이메일 국가 제품 수 이점
TargetMol Chemicals Inc.
+1-781-999-5354 +1-00000000000
marketing@targetmol.com United States 19892 58
3B Pharmachem (Wuhan) International Co.,Ltd. 821-50328103-801 18930552037
3bsc@sina.com China 15848 69
EMMX Biotechnology LLC 888-539-0666
info@emmx.com United States 8449 60
TargetMol Chemicals Inc. 4008200310
marketing@tsbiochem.com China 24131 58
ApexBio Technology --
sales@apexbt.com United States 6254 58

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