4-BENZYL-2-METHYL-1,2,4-THIADIAZOLIDINE-3,5-DIONE C화학적 특성, 용도, 생산
화학적 성질
White Solid
용도
Glycogen Synthase Kinase-3? is a highly conserved ubiquitously expressed serine/threonine protein kinase involved in signal transduction cascades of multiple cellular processes. TDZD-8 is a thiadiazolidinone (TDZD) analogue that acts as a highly selectiv
일반 설명
A cell-permeable, thiadiazolidinone (TDZD) analog that acts as a highly selective, non-ATP-competitive inhibitor of GSK-3β (IC50 = 2 μM). Inhibits Flt-3 and PKC activities (IC50 = 673 nM and 1.4-5.5 μM, respectively). Does not significantly affect the activities of Cdk1/cyclin B, CK-II, PKA, or PKC (IC50 >100 μM). Shown to inhibit collagen- and thrombin-induced platelet aggregation.
4-BENZYL-2-METHYL-1,2,4-THIADIAZOLIDINE-3,5-DIONE 준비 용품 및 원자재
원자재
준비 용품
4-BENZYL-2-METHYL-1,2,4-THIADIAZOLIDINE-3,5-DIONE 공급 업체