Company Name: |
Shanghai Hongye Biotechnology Co. Ltd
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Tel: |
400-9205774 |
Email: |
sales@glpbio.cn |
Products Intro: |
Product Name:Amauromine CAS:88360-87-6 Purity:>98% Package:1mg;10mg;50mg;100mg;
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Company Name: |
Energy Chemical
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Tel: |
021-58432009 400-005-6266 |
Email: |
marketing@energy-chemical.com |
Products Intro: |
Product Name:Amauromine CAS:88360-87-6 Purity:NULL Package:1mg;2.5mg Remarks:NULL
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| amauromine Basic information |
Product Name: | amauromine | Synonyms: | amauromine;(5aS)-8aα,16aα-Bis(1,1-dimethyl-2-propenyl)-5aα,8,8a,13,13aα,15aβ,16,16a-octahydropyrazino[1'',2'':1,5:4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aβH)-dione;Antibiotic FR-900220;FR-900220;WF-6237;(5aS,7aS,8aR,13aS,15aS,16aR)-8a,16a-Bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-pyrazino[1'',2'':1,5;4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione;4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione, 8a,16a-bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-, (5aS,7aS,8aR,13aS,15aS,16aR)- | CAS: | 88360-87-6 | MF: | C32H36N4O2 | MW: | 508.662 | EINECS: | | Product Categories: | | Mol File: | 88360-87-6.mol | |
| amauromine Chemical Properties |
Boiling point | 689.9±55.0 °C(Predicted) | density | 1.28±0.1 g/cm3(Predicted) | storage temp. | Store at -20°C | solubility | DMSO: Soluble; Ethanol: Soluble; Methanol: Soluble | form | A solid | pka | 3.26±0.60(Predicted) | color | Brown |
Toxicity | LD50 intraperitoneal in mouse: > 200mg/kg |
| amauromine Usage And Synthesis |
Description | Amauromine is a neutral antagonist of the cannabinoid (CB) receptor CB1 that is selective for CB1 (Ki = 178 nM; Kb = 66.6 nM) over CB2, with no activity at CB2 receptors at concentrations up to 10 μM. It is also an antagonist of GPR18 (IC50 = 3.74 μM). Amauromine has vasodilatory activity. | Uses | Amauromine is a CB1 and Calcium Channel antagonist. | storage | +4°C |
| amauromine Preparation Products And Raw materials |
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