STILBAMIDINE
| 中文名称 | STILBAMIDINE |
|---|---|
| 中文同义词 | 司替巴脒;化合物 T13905 |
| 英文名称 | stilbamidine |
| 英文同义词 | stilbamidine;4,4'-Stilbenedicarboxamidine;2-(2-phenylethenyl)benzenecarboximidamide;Ba 2652;Stilbamidin;Benzenecarboximidamide, 4,4'-(1,2-ethenediyl)bis- |
| CAS号 | 122-06-5 |
| 分子式 | C16H16N4 |
| 分子量 | 264.33 |
| EINECS号 | 2045195 |
| 相关类别 | |
| Mol文件 | 122-06-5.mol |
| 结构式 |  |
STILBAMIDINE 性质
| 沸点 | 397.56°C (rough estimate) |
|---|---|
| 密度 | 1.1536 (rough estimate) |
| 折射率 | 1.6000 (estimate) |
| 储存条件 | Store at -20°C |
| 溶解度 | 溶于二甲基亚砜 |
fungal
The high-affinity pentamidine transporter (HAPT1) is inhibited by Propamidine but displays only low affinity to Stilbamidine. adenosine-sensitive pentamidine transporter (ASPT1), in contrast, is strongly inhibited by Stilbamidine, and Propamidine. [ 3 H]pentamidine uptake is determined in the presence of various concentrations of adenosine (IC 50 =1.2 μM) or melarsen oxide (IC 50 =0.7 μM), as well as in the presence of 250 μM adenosine and increasing concentrations of hypoxanthine, Propamidine (IC 50 =6.1 μM) and Stilbamidine (IC 50 =110 μM). The two diamidine compounds, Stilbamidine and Pentamidine are used to treat in multiple myeloma, a disease in which increase of the globulin content of the serum is of frequent occurrence.
安全信息
| 更新日期 | 产品编号 | 产品名称 | CAS号 | 包装 | 价格 |
|---|---|---|---|---|---|
| 2023/03/20 | HY-U00007 | STILBAMIDINE Stilbamidine | 122-06-5 | 5mg | 6200元 |