(D(CH2)51,TYR(ET)2,VAL4,ARG8)-VASOPRESSIN
| 中文名称 | (D(CH2)51,TYR(ET)2,VAL4,ARG8)-VASOPRESSIN |
|---|---|
| 中文同义词 | |
| 英文名称 | BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENE-PROPIONYL-TYR(ET)-PHE-VAL-ASN-CYS-PRO-ARG-GLY-NH2 |
| 英文同义词 | (B-MERCAPTO-B,B-CYCLOPENTAMETHYLENE-*PRO PIONYL1,O-E;[β-mercapto-β,β-cyclopentamethylenepropionyl1, o-et-tyr2, val4, arg8]-vasopressin;1-(1-MERCAPTOCYCLOHEXANEACETIC ACID)-2-(O-ETHYL-L-TYROSINE)-4-L- VALINE-8-L-ARGININEVASOPRESSIN;vasopressin 1-(1-MCHA)-2-(O-ethyl-L-tyrosine)-4-L-valine;BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENE-PROPIONYL-TYR(ET)-PHE-VAL-ASN-CYS-PRO-ARG-GLY-NH2;[BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENEPROPIONYL1,O-ET-TYR2,VAL4,ARG8]-VASOPRESSIN;(D(CH2)(5/1),TYR(ET)2,VAL4,ARG8)-VASOPRESSIN;[1-MERCAPTOCYCLOHEXYL]ACETYL-TYR[O-ETHYL]-PHE-VAL-ASN-CYS-PRO-ARG-GLY-NH2 |
| CAS号 | 77453-01-1 |
| 分子式 | C53H77N13O11S2 |
| 分子量 | 1136.39 |
| EINECS号 | |
| 相关类别 | Vasopressin and Oxytocin receptor;Hormones;Oxytocin&Vasopressin;Pituitary Hormones;VasopressinPeptides for Cell Biology;Vasopressins |
| Mol文件 | 77453-01-1.mol |
| 结构式 |  |
(D(CH2)51,TYR(ET)2,VAL4,ARG8)-VASOPRESSIN 性质
| 储存条件 | −20°C |
|---|
SKF 100398 (d(CH2)5Tyr(Et)VAVP) 是一种精氨酸加压素 (AVP) 类似物，能作为外源性和内源性 AVP 抗利尿作用的特异性拮抗剂。
SKF 100398 is a specific antagonist of the hydrosmotic effect of exogenous and endogenous AVP.
SKF 100398 (8 μg/kg; i.v.) abolishes the antidiuretic effect of AVP.
| Animal Model: | Male Sprague-Dawley rats (250-300 g) |
| Dosage: | 8 μg/kg |
| Administration: | Intravenous injection |
| Result: | Completely blocked the antidiuretic effect of exogenous AVP (4 ng/kg body wt i.v.). |
| 提供商 | 语言 |
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英文
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