Clopidogrel thiolactone NEW
| Price | $228 |
| Package | 5mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-11-04 |
Product Details
| Product Name: Clopidogrel thiolactone | CAS No.: 1147350-75-1 |
| Purity: 98.79% | Supply Ability: 10g |
| Release date: 2025/11/04 |
Product Introduction
Bioactivity
| Name | Clopidogrel thiolactone |
| Description | Clopidogrel thiolactone (2-oxoclopidogrel) is a potent P2Y12 receptor inhibitor and a potent antiplatelet aggregation compound.Clopidogrel thiolactone is the active metabolic intermediate resulting from the first oxidative activation of Clopidogrel. |
| In vivo | Clopidogrel thiolactone holds great promise as a more potent and a safer antiplatelet agent that might have the following advantages over clopidogrel: (1) no drug resistance for CYP2C19 poor metabolizers; (2) lower dose-related toxicity due to a much lower effective dose; (3) faster onset of action. Clopidogrel thiolactone (8 μm/kg; i.v.; Sprague-Dawley male rats) exhibits good biological availability and pharmacokinetic parameters[2]. |
| Storage | store at low temperature,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Solubility Information | 10% DMSO+40% PEG300+5% Tween 80+45% Saline : 2 mg/mL (5.92 mM), Sonication is recommended. Ethanol : 2 mg/mL (5.92 mM), Sonication and heating are recommended. DMSO : 30 mg/mL (88.80 mM), Sonication is recommended. |
| Keywords | P2YReceptor | P2Y12 | P2Y Receptor | Clopidogrel thiolactone |
| Inhibitors Related | Melamine | Mycophenolate Mofetil | Clozapine N-Oxide | L-Threonic acid magnesium salt | Isonicotinic acid | Uridine-5'-diphosphate disodium salt | Urolithin A | Lansoprazole sulfide | Tulipalin A | 4-(4-Amino-3-fluorophenoxy)-N-methylpicolinamide | Nicotinamide N-oxide | Ticagrelor |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, USA
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