Immunoproteasome inhibitor 1 NEW
| Price | $1520 | $1980 | $2500 |
| Package | 25mg | 50mg | 100mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-10-27 |
Product Details
| Product Name: Immunoproteasome inhibitor 1 | CAS No.: 2755772-63-3 |
| Supply Ability: 10g | Release date: 2025/10/27 |
Product Introduction
Bioactivity
| Name | Immunoproteasome inhibitor 1 |
| Description | Immunoproteasome inhibitor 1 is a highly potent and reversible inhibitor of both immunoproteasome and proteasome activity. It exhibits time-independent inhibitory effects on immunoproteasome subunits β5c, β1i, and β5i, with respective Ki values of 1.18 μM, 0.27 μM, and 1.91 μM. This compound shows promising potential for the treatment of select neoplastic diseases [1]. |
| In vitro | Immunoproteasome inhibitor 1 (compound 9), used in concentrations ranging from 0 to 25 μM for durations of 0 to 600 seconds in Human 20S immunoproteasome and human 20S proteasome, exhibits a high binding affinity, particularly for the β1i subunit (0.27 μM). Additionally, it demonstrates effective inhibition of both β5i and β5c subunits. Notably, inhibition of the β5i subunit is characterized as reversible and independent of exposure time [1]. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Inhibitors Related | MG-132 | Tripterin | Sitagliptin | Teneligliptin hydrobromide | Carfilzomib | Sitagliptin phosphate monohydrate | Anagliptin | Linagliptin | Vildagliptin | Alloxan monohydrate | 4'-Hydroxychalcone | Bortezomib |
Company Profile Introduction
TargetMol Chemicals Inc. is headquartered in Boston, MA, and specializes in products and services that serve the research needs of chemical and biological scientists worldwide. With a client base in 40+ countries, TargetMol has evolved into one of the biggest global research suppliers for compound libraries and small molecule compounds.
170+ Compound Libraries， 10000+ Noval Small Molecucles，16000+ Nature Compounds
TargetMol diligently updates and offers over 170 types of compound libraries and a wide range of high-quality research chemicals, including inhibitors, activators, natural products, peptides, antibodies , and novel life-science kits for laboratory and scientific use. In addition, our lab allows us to conduct CADD (computer-aided drug design) and chemical synthesis to meet the customization needs of our clients.
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- Address: 36 Washington Street, Wellesley Hill, Massachusetts, USA
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