PKM2 activator 3 NEW
| Price | $1520 | $1980 | $2500 |
| Package | 25mg | 50mg | 100mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-10-27 |
Product Details
| Product Name: PKM2 activator 3 | CAS No.: 1346113-84-5 |
| Supply Ability: 10g | Release date: 2025/10/27 |
Product Introduction
Bioactivity
| Name | PKM2 activator 3 |
| Description | PKM2 activator 3 is a highly potent compound that activates PKM2, with an AC 50 value of 90 nM. It exhibits excellent Caco-2 permeability, a low efflux ratio, and remarkable microsomal stability. PKM2 activator 3 is particularly valuable for anticancer research purposes [1]. (AC 50: the concentration at which 50% enzyme activation occurs.) |
| In vivo | PKM2 activator 3, also known as compound 66, exhibits favorable pharmacokinetic properties, including efficient Caco-2 permeability and a low efflux ratio of 0.84. It demonstrates robust microsomal stability, with a half-life of 277.2 minutes in human liver microsomes and 117.5 minutes in mouse liver microsomes [1]. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Inhibitors Related | DL-Serine | PKM2-IN-1 | PKR-IN-2 | Disodium monofluorophosphate | Mitapivat | (+)-Shikonin | PKM2 inhibitor G | DASA-58 | Dimethylaminomicheliolide HCl | TEPP-46 | Mitapivat sulfate hydrate | PKM2 activator 2 |
Company Profile Introduction
TargetMol Chemicals Inc. is headquartered in Boston, MA, and specializes in products and services that serve the research needs of chemical and biological scientists worldwide. With a client base in 40+ countries, TargetMol has evolved into one of the biggest global research suppliers for compound libraries and small molecule compounds.
170+ Compound Libraries， 10000+ Noval Small Molecucles，16000+ Nature Compounds
TargetMol diligently updates and offers over 170 types of compound libraries and a wide range of high-quality research chemicals, including inhibitors, activators, natural products, peptides, antibodies , and novel life-science kits for laboratory and scientific use. In addition, our lab allows us to conduct CADD (computer-aided drug design) and chemical synthesis to meet the customization needs of our clients.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, Massachusetts, USA
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