Bayer-18
|
N-叔丁基-N'-[3-[[5-氟-4-[(2-羟基-1,1-二甲基乙基)氨基]-2-嘧啶基]氨基]苯基]脲
|
1251752-12-1
|
BEZ235
|
NVP-BEZ235
|
915019-65-7
|
BI-2536
|
BI 2536
|
755038-02-9
|
BI-D1870
|
BI-D1870
|
501437-28-1
|
BisindolylMaleiMide X, HCl salt
|
RO 31-8425
|
1241725-87-0
|
BMS-2
|
1-(4-氟苯基)-N-[3-氟-4-(1H-吡咯并[2,3-B]吡啶-4-基氧基)苯基]-1,2-二氢-2-氧代-3-吡啶甲酰胺
|
888719-03-7
|
BMS-3
|
|
|
BMS-5
|
|
|
BMS-599626
|
AC480 (BMS-599626)
|
714971-09-2
|
Brivanib
|
酪氨酸激酶抑制剂
|
649735-46-6
|
Brivanib alaninate
|
1-[[4-[(4-氟-2-甲基-1H-吲哚-5-基)氧基]-5-甲基吡咯并[2,1-F][1,2,4]三嗪-6-基]氧基]-2-丙醇 L-丙氨酸酯
|
649735-63-7
|
BS194
|
(2S,3S)-3-[[3-(异丙基)-7-[(苯基甲基)氨基]吡唑并[1,5-A]嘧啶-5-基]氨基]-1,2,4-丁三醇
|
1092443-55-4
|
BX-795
|
N-[3-[[5-碘-4-[[3-[(2-噻吩基羰基)氨基]丙基]氨基]-2-嘧啶基]氨基]苯基]-1-吡咯烷甲酰胺
|
702675-74-9
|
BX-912
|
BX-912
|
702674-56-4
|
Cabozantinib
|
卡博替尼
|
849217-68-1
|
Canertinib
|
卡奈替尼
|
267243-28-7
|
CC-401
|
3-[3-[2-(1-哌啶基)乙氧基]苯基]-5-(1H-1,2,4-三唑-5-基)-1H-吲唑
|
395104-30-0
|
CEP-33779
|
N-[3-(4-甲基-1-哌嗪基)苯基]-8-[4-(甲磺酰基)苯基]-[1,2,4]三唑并[1,5-A]吡啶-2-胺
|
1346168-57-7
|
CH5132799
|
CH5132799
|
1007207-67-1
|
CI-1040
|
2-[(2-氯-4-碘苯基)氨基]-N-(环丙基甲氧基)-3,4-二氟-苯甲酰胺
|
212631-79-3
|
CP-724714
|
2-甲氧基-N-[(2E)-3-[4-[[3-甲基-4-[(6-甲基-3-吡啶基)氧基]苯基]氨基]-6-喹唑啉基]-2-丙烯-1-基]乙酰胺
|
383432-38-0
|
Crizotinib
|
克唑替尼
|
877399-52-5
|
CX-4945
|
CX-4945
|
1009820-21-6
|
CYC-116
|
CYC-116
|
693228-63-6
|
Danusertib
|
达鲁舍替
|
827318-97-8
|
Dasatinib
|
达沙替尼
|
302962-49-8
|
DianilinopyriMidine_01
|
N2-(4-(氨甲基)苯)-5-氟-N4-苯基嘧啶-2,4-二胺
|
916603-07-1
|
diethyl 7-oxo-4,7-dihydropyrazolo[1,5-a]pyriMidine-3,6-dicarboxylate
|
7-氧代-4,7-二氢吡唑并[1,5-A]-嘧啶-3,6-二羧酸二乙酯
|
155374-25-7
|
Dovitinib
|
4-氨基-5-氟-3-[5-(4-甲基哌嗪-1-基)-1H-苯并咪唑-2-基]喹啉-2(1H)-酮
|
405169-16-6
|
E7080
|
乐伐替尼
|
417716-92-8
|
Erlotinib Hydrochloride
|
盐酸埃罗替尼
|
183319-69-9
|
ethyl 2-(Methylthio)-4-oxo-3,4-dihydropyrazolo[1,5-a][1,3,5]triazine-8-carboxylate
|
|
278600-53-6
|
ethyl 3-aMinofuro[2,3-b]pyridine-2-carboxylate
|
3-氨基-呋喃并[2,3-B]嘧啶-2-甲酸乙酯
|
371945-06-1
|
ethyl 3-aMinothieno[2,3-b]pyridine-2-carboxylate
|
3-氨基噻吩并[2,3-B]吡啶-2-甲酸乙酯
|
52505-46-1
|
ethyl 3-cyano-7-oxo-4,7-dihydropyrazolo[1,5-a]pyriMidine-6-carboxylate
|
3-氰基-7-氧代-4,7-二氢吡唑并[1,5-A]嘧啶-6-羧酸乙酯
|
64689-83-4
|
ethyl 5-chloropyrazolo[1,5-a]pyriMidine-3-carboxylate
|
5-氯吡唑并[1,5-a]嘧啶-3-羧酸乙酯
|
1224944-77-7
|
ethyl 5-oxo-4,5-dihydropyrazolo[1,5-a]pyriMidine-3-carboxylate
|
5-氧代-4,5-二氢吡唑并[1,5-a]嘧啶-3-羧酸乙酯
|
926663-00-5
|
ethyl 7-aMino-5-hydroxypyrazolo[1,5-a]pyriMidine-3-carboxylate
|
7-氨基-5-氧代-4,5-二氢吡唑并[1,5-A]嘧啶-3-羧酸乙酯
|
90674-09-2
|
ethyl 7-aMinopyrazolo[1,5-a]pyriMidine-3-carboxylate
|
7-氨基吡唑并[1,5-A]嘧啶-3-羧酸乙酯
|
1196153-97-5
|
ethyl 7-chloropyrazolo[1,5-a]pyriMidine-3-carboxylate
|
乙基 7-氯吡唑并[1,5-A]嘧啶-3-甲酸基酯
|
749216-54-4
|
ethyl 7-oxo-4,7-dihydropyrazolo[1,5-a]pyriMidine-3-carboxylate
|
7-氧代-4,7-二氢吡唑并[1,5-A]嘧啶-3-羧酸乙酯
|
104556-86-7
|
ethyl pyrazolo[1,5-a]pyriMidine-3-carboxylate
|
吡唑并[1,5-A]嘧啶-3-羧酸乙酯
|
115932-00-8
|
GDC-0941
|
GDC-0941
|
957054-30-7
|
GDC0980
|
(S)-1-[4-[[2-(2-氨基嘧啶-5-基)-7-甲基-4-(吗啉-4-基)噻吩并[3,2-D]嘧啶-6-基]甲基]哌嗪-1-基]-2-羟基丙-1-酮
|
1032754-93-0
|
Gefitinib
|
吉非替尼
|
184475-35-2
|
GNE 477
|
GNE 477
|
1032754-81-6
|
GNE-490
|
2-(2-氨基-4-甲基-5-嘧啶基)-ALPHA,ALPHA-二甲基-4-(4-吗啉基)噻吩并[3,2-D]嘧啶-6-甲醇
|
1033739-92-2
|
GNE-493
|
GNE-493
|
1033735-94-2
|
GPLG0634
|
非戈替尼
|
1206161-97-8
|
GSK2126458
|
GSK2126458
|
1086062-66-9
|
GSK-25
|
GSK-25
|
874119-56-9
|
GSK690693
|
4-[2-(4-氨基-1,2,5-恶二唑-3-基)-1-乙基-7-[(3S)-3-哌啶基甲氧基]-1H-咪唑并[4,5-C]吡啶-4-基]-2-甲基-3-丁炔-2-醇
|
937174-76-0
|
GW441756
|
GW441756
|
504433-23-2
|
IC87114
|
2-[(6-氨基-9H-嘌呤-9-基)甲基]-5-甲基-3-(2-甲基苯基)-4(3H)-喹唑啉酮
|
371242-69-2
|
IMatinib Mesylate
|
甲磺酸伊马替尼
|
221027-57-1
|
INK128
|
3-(2-氨基-5-苯并恶唑基)-1-(1-甲基乙基)-1H-吡唑并[3,4-D]嘧啶-4-胺
|
1224844-38-5
|
Intedanib
|
尼达尼布
|
656247-17-5
|
isoxazolo[5,4-b]pyridin-3-aMine
|
异恶唑并[5,4-B]吡啶-3-胺
|
92914-74-4
|
JNJ-28312141
|
4-CYANO-N-[2-(CYCLOHEX-1-EN-1-YL)-4-{1-[2-(DIMETHYLAMINO)ACETYL]PIPERIDIN-4-YL}PHENYL]-1H-IMIDAZOLE-2-CARBOXAMIDE
|
885692-52-4
|
JNJ-38158471
|
CS-2660
|
951151-97-6
|
JNJ38877605
|
6-[二氟[6-(1-甲基-1H-吡唑-4-基)-1,2,4-噻唑并[4,3-B]吡嗪-3-基]甲基]-喹啉
|
943540-75-8
|
JNJ7706621
|
JNJ-7706621
|
443797-96-4
|
Ki20227
|
Ki20227
|
623142-96-1
|
KU0063794
|
KU-0063794
|
938440-64-3
|
KU55933
|
2-吗啉-4-基-6-噻蒽-1-基吡喃-4-酮
|
587871-26-9
|
KU57788
|
8-(4-二苯并噻吩基)-2-(4-吗啉基)-4H-1-苯并吡喃-4-酮
|
503468-95-9
|
Lapatinib
|
拉帕替尼
|
231277-92-2
|
Linifanib
|
利尼伐尼
|
796967-16-3
|
LY294002
|
LY294002/PI3K抑制剂
|
154447-36-6
|
Masatinib
|
马赛替尼(Masitinib)
|
790299-79-5
|
Merck-22-6
|
Merck-22-6
|
12847-42-4
|
Merck-5
|
2-(1,1-二甲基乙基)-9-氟-1,6-二氢-7H-苯并[H]咪唑并[4,5-F]异喹啉-7-酮
|
457081-03-7
|
MK-2461
|
MK-2461
|
917879-39-1
|
MoMelotinib
|
莫洛替尼
|
1056634-68-4
|
Motesanib
|
莫特塞尼
|
453562-69-1
|
Mubritinib
|
木利替尼
|
366017-09-6
|
Neratinib
|
来那替尼
|
698387-09-6
|
NIBR-17
|
CS-2663
|
944396-88-7
|
Nilotinib
|
尼罗替尼
|
641571-10-0
|
NVP-BGJ398
|
FGFR抑制剂(NVP-BGJ398)
|
872511-34-7
|
NVP-BSK805
|
NVP-BSK805 dihydrochloride
|
1092499-93-8
|
Pazopanib
|
帕唑帕尼
|
444731-52-6
|
Pazopanib HCl
|
盐酸帕唑帕尼
|
635702-64-6
|
PD0325901
|
N-[(2R)-2,3-二羟基丙氧基]-3,4-二氟-2-[(2-氟-4-碘苯)氨基]苯甲酰胺
|
391210-10-9
|
PD173955
|
6-(2,6-二氯苯基)-8-甲基-2-[[3-(甲硫基)苯基]氨基]吡啶并[2,3-D]嘧啶-7(8H)-酮
|
260415-63-2
|
PD173955-Analog 1
|
3-[[6-(2,6-二氯苯基)-7,8-二氢-8-甲基-7-氧代吡啶并[2,3-D]嘧啶-2-基]氨基]苯甲酸
|
185039-99-0
|
Pelitinib
|
培利替尼
|
257933-82-7
|
PF04217903
|
2-[4-[1-(喹啉-6-甲基)-1H-[1,2,3]三唑并[4,5-B]吡嗪-6-基]-1H-吡唑-1-基]乙醇
|
956905-27-4
|
PF431396
|
N-甲基-N-[2-[[[2-[(2-氧代-2,3-二氢-1H-吲哚-5-基)氨基]-5-三氟甲基嘧啶-4-基]氨基]甲基]苯基]甲磺酰胺
|
717906-29-1
|
PF-562271
|
N-甲基-N-[3-[[[2-[(2-氧代-2,3-二氢-1H-吲哚-5-基)氨基]-5-三氟甲基嘧啶-4-基]氨基]甲基]吡啶-2-基]甲磺酰胺
|
717907-75-0
|
PHA690509
|
(2S)-2-[4-(乙酰基氨基)苯基]-N-(5-异丙基噻唑-2-基)丙酰胺
|
492445-28-0
|
PI-103
|
PI-103
|
371935-74-9
|
PIK-294
|
PIK-294
|
900185-02-6
|
PIK-75
|
2-甲基-5-硝基-1-苯磺酰[2-[(6-溴咪唑并[1,2-A]吡啶-3-基)亚甲基]-1-甲基肼]
|
372196-67-3
|
PIK-90
|
N-(2,3-二氢-7,8-二甲氧基咪唑并[1,2-C]喹唑啉-5-基)-3-吡啶甲酰胺
|
677338-12-4
|
PIK-93
|
N-[5-[4-氯-3-[[(2-羟基乙基)氨基]磺酰基]苯基]-4-甲基-2-噻唑基]乙酰胺
|
593960-11-3
|
PLX4720
|
N-[3-[(5-氯-1H-吡咯并[2,3-B]吡啶-3-基)羰基]-2,4-二氟苯基]-1-丙磺酰胺
|
918505-84-7
|
Ponatinib
|
帕纳替尼
|
943319-70-8
|
Purvalanol B
|
(2R)-2-[[6-[(3-氯-4-羧基苯基)氨基]-9-(1-甲基乙基)-9H-嘌呤-2-基]氨基]-3-甲基-1-丁醇
|
212844-54-7
|
pyrazolo[1,5-a][1,3,5]triazine-2,4-diol
|
吡唑并[1,5-A]-1,3,5-三嗪-2,4(1H,3H)-二酮
|
34683-40-4
|