Butabindide oxalate

Butabindide oxalate Struktur
185213-03-0
CAS-Nr.
185213-03-0
Englisch Name:
Butabindide oxalate
Synonyma:
[S-(R*,R*)]-1-(2-Amino-1-oxobutyl)-N-butyl-2,3-dihydro-1H-indole-2-carboxamide ethanedioate
CBNumber:
CB12597437
Summenformel:
C19H27N3O6
Molgewicht:
393.43418
MOL-Datei:
185213-03-0.mol

Butabindide oxalate Eigenschaften

Schmelzpunkt:
142 °C
storage temp. 
Desiccate at -20°C
Löslichkeit
Soluble to 100 mM in water and to 100 mM in DMSO
Aggregatzustand
Powder

Sicherheit

Butabindide oxalate Chemische Eigenschaften,Einsatz,Produktion Methoden

Beschreibung

Butabindide is a potent inhibitor of cholecystokinin-inactivating peptidase/tripeptidyl peptidase 2 (CCK-inactivating peptidase/TPP-2; Ki = 7 nM). It is selective for CCK-inactivating peptidase/TPP-2 over a panel of serine proteases (Kis = >1 μM) as well as CCK receptors (Kis = >0.1 mM). Butabindide (0.1-100 μM) increases levels of CCK octapeptide (Item Nos. 24404 | 23371) in depolarized rat cerebral cortex slices. In vivo, butabindide inhibits CCK-inactivating peptidase/TPP-2 in mouse liver and brain (ID50s = 1.1 and 6.8 mg/kg, respectively). It also enhances CCK octapeptide-induced delay in gastric emptying and reduces food intake in mice.

Butabindide oxalate Upstream-Materialien And Downstream Produkte

Upstream-Materialien

Downstream Produkte


Butabindide oxalate Anbieter Lieferant Produzent Hersteller Vertrieb Händler.

Global( 19)Lieferanten
Firmenname Telefon E-Mail Land Produktkatalog Edge Rate
TargetMol Chemicals Inc.
+1-781-999-5354 +1-00000000000
marketing@targetmol.com United States 19892 58
Aladdin Scientific
+1-833-552-7181
sales@aladdinsci.com United States 52927 58
VDM Biochemicals 0330-2528181
sales@vdmbio.com United States 510 64
Shanghai EFE Biological Technology Co., Ltd. 021-65675885 18964387627
info@efebio.com China 9709 58
Amatek Scientific Co. Ltd. 0512-56316828
info@amateksci.com China 28821 58
BOC Sciences --
info@bocsci.com USA 0 65
DC Chemicals 021-58447131 13564518121
sales@dcchemicals.com China 9414 58
MedBioPharmaceutical Technology Inc 021-69568360 18916172912
order@med-bio.cn China 8141 58
Changzhou Furuisi Biotechnology Co., Ltd 0519-85524369
3477467573@qq.com China 8618 58
TargetMol Chemicals Inc. 4008200310
marketing@tsbiochem.com China 24018 58

  • [S-(R*,R*)]-1-(2-Amino-1-oxobutyl)-N-butyl-2,3-dihydro-1H-indole-2-carboxamide ethanedioate
  • 185213-03-0
  • Inhibitor of tripeptidyl peptidase II (TPPII).
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