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NALTRIBEN MESYLATE

CAS No.
111555-58-9
Chemical Name:
NALTRIBEN MESYLATE
Synonyms
NTB;NALTRIBEN MESYLATE;naltrindolebenzofuran;NALTRIBEN METHANESULFONATE;17-(Cyclopropylmethyl)-6,7-didehydro-3,14β-dihydroxy-4,5α-epoxy-6,7-2',3'-benzo[b]furanomorphinanmesylate;17-(Cyclopropylmethyl)-6,7-didehydro-3,14b-dihydroxy-4,5a-epoxy-6,7-2',3'-benzo[b]furanomorphinanmesylate;17-(CYCLOPROPYLMETHYL)-6,7-DIDEHYDRO-3, 14B-DIHYDROXY-4,5A-EPOXY-6,7-2',3'-BENZO[B]FURANOMORPHINAN MESYLATE;17-(Cyclopropylmethyl)-6,7-didehydro-3-4,5alpha-epoxy-14beta-dihydroxy-6,7-2',3'-benzo[b]furanomorphinan mesylate;4,8-Methano-8aH-bisbenzofuro[3,2-e:2',3'-g]isoquinoline-1,8a-diol, 7-(cyclopropylmethyl)-5,6,7,8,9,14b-hexahydro-, (4bS,8R,8aS,14bR)-
CBNumber:
CB2112297
Molecular Formula:
C26H25NO4
Molecular Weight:
415.48
MDL Number:
MFCD00673953
MOL File:
111555-58-9.mol
Last updated:2023-05-04 17:34:31

NALTRIBEN MESYLATE Properties

Boiling point 605.3±55.0 °C(Predicted)
Density 1.50±0.1 g/cm3(Predicted)
storage temp. −20°C
solubility DMSO: 14 mg/mL at ~60 °C
form solid
pka 9.30±0.40(Predicted)
color off-white
FDA UNII RXG719F189

SAFETY

Risk and Safety Statements

WGK Germany  3
RTECS  PB9175000

NALTRIBEN MESYLATE price More Price(7)

Manufacturer Product number Product description CAS number Packaging Price Updated Buy
Usbiological 460532 Naltriben Mesylate 111555-58-9 1mg $382 2021-12-16 Buy
TRC N284430 Naltriben 111555-58-9 50mg $795 2021-12-16 Buy
Biosynth Carbosynth FN73528 Naltriben 111555-58-9 10mg $125 2021-12-16 Buy
AK Scientific 1744CP Naltriben 111555-58-9 10mg $218 2021-12-16 Buy
Biosynth Carbosynth FN73528 Naltriben 111555-58-9 50mg $437.5 2021-12-16 Buy
Product number Packaging Price Buy
460532 1mg $382 Buy
N284430 50mg $795 Buy
FN73528 10mg $125 Buy
1744CP 10mg $218 Buy
FN73528 50mg $437.5 Buy

NALTRIBEN MESYLATE Chemical Properties,Uses,Production

Uses

Naltriben is a potent and selective antagonist for the δ2 opioid receptor. Naltriben is used to differentiate the δ1 and δ2 opioid receptors.

Definition

ChEBI: Naltriben is a morphinane alkaloid.

Biological Activity

Selective and potent δ -opioid receptor antagonist (K i values are 0.013, 19 and 152 nM for δ , μ and κ receptors respectively). Displays selectivity for the δ 2 subtype in vivo .

NALTRIBEN MESYLATE Preparation Products And Raw materials

Raw materials

Preparation Products

NALTRIBEN MESYLATE Suppliers

Global( 21)Suppliers
Supplier Tel Email Country ProdList Advantage
3B Pharmachem (Wuhan) International Co.,Ltd. 821-50328103-801 18930552037 3bsc@sina.com China 15848 69
EMMX Biotechnology LLC 888-539-0666 info@emmx.com United States 8449 60
Shanghai Universal Biotech Co.,Ltd 18768175414 gaojun@univ-bio.com China 24998 58
Carbosynth -- sales@carbosynth.com United Kingdom 6018 58
NTB NALTRIBEN MESYLATE NALTRIBEN METHANESULFONATE naltrindolebenzofuran 17-(Cyclopropylmethyl)-6,7-didehydro-3-4,5alpha-epoxy-14beta-dihydroxy-6,7-2',3'-benzo[b]furanomorphinan mesylate 17-(Cyclopropylmethyl)-6,7-didehydro-3,14β-dihydroxy-4,5α-epoxy-6,7-2',3'-benzo[b]furanomorphinanmesylate 17-(CYCLOPROPYLMETHYL)-6,7-DIDEHYDRO-3, 14B-DIHYDROXY-4,5A-EPOXY-6,7-2',3'-BENZO[B]FURANOMORPHINAN MESYLATE 17-(Cyclopropylmethyl)-6,7-didehydro-3,14b-dihydroxy-4,5a-epoxy-6,7-2',3'-benzo[b]furanomorphinanmesylate 4,8-Methano-8aH-bisbenzofuro[3,2-e:2',3'-g]isoquinoline-1,8a-diol, 7-(cyclopropylmethyl)-5,6,7,8,9,14b-hexahydro-, (4bS,8R,8aS,14bR)- 111555-58-9 C26H25NO4CH3SO3H C27H29NO7S Opioid receptor and opioid-like receptor