(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE

(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE C화학적 특성, 용도, 생산

생물학적 활성

Potent and selective antagonist for the human adenosine A 3 receptor, with low affinity for the rat A 3 receptor (K i values are 2.3 and > 10000 nM respectively). Displays > 1000-fold selectivity over human A 1 and A 2A receptors (K i values are 4.1 and 3.3 μ M respectively) and > 180-fold selectivity over rat A 1 , rat A 2A and mouse A 2B receptors. Acts as an inverse agonist in the [ 35 S]GTP γ S binding assay in hA 3 -CHO cells (IC 50 = 36 nM).

(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE 준비 용품 및 원자재

원자재

준비 용품

(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE 공급 업체

공급자	전화	이메일	국가	제품 수	이점
3B Pharmachem (Wuhan) International Co.,Ltd.	821-50328103-801 18930552037	3bsc@sina.com	China	15848	69
EMMX Biotechnology LLC	888-539-0666	info@emmx.com	United States	8449	60
United States Biological	--	sales@advtechind.com	United States	6106	58

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