(2S)-1-[[(2R,3S)-5-CHLORO-3-(2-CHLOROPHENYL)-1-[(3,4-DIMETHOXYPHENYL)SULFONYL]-2,3-DIHYDRO-3-HYDROXY-1H-INDOL-2-YL]CARBONYL]-2-PYRROLIDINECARBOXAMIDE
- $49 - $3200
- Product name: (2S)-1-[[(2R,3S)-5-CHLORO-3-(2-CHLOROPHENYL)-1-[(3,4-DIMETHOXYPHENYL)SULFONYL]-2,3-DIHYDRO-3-HYDROXY-1H-INDOL-2-YL]CARBONYL]-2-PYRROLIDINECARBOXAMIDE
- CAS: 150375-75-0
- MF: C28H27Cl2N3O7S
- MW: 620.5
- EINECS:
- MDL Number:MFCD00922133
- Synonyms:(2S)-1-[[(2R,3S)-5-CHLORO-3-(2-CHLOROPHENYL)-1-[(3,4-DIMETHOXYPHENYL)SULFONYL]-2,3-DIHYDRO-3-HYDROXY-1H-INDOL-2-YL]CARBONYL]-2-PYRROLIDINECARBOXAMIDE;INDOL-2-YLCARBONYL)-L-PROLINAMIDE;Relcovaptan;reclovaptan;SR 49059;Relcovaptan (SR-49059);2-Pyrrolidinecarboxamide, 1-[[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-, (2S)-
23 prices
Selected condition:
Brand
- aablocks
- ACHEMBLOCK
- AHH
- AK Scientific
- American Custom Chemicals Corporation
- ApexBio Technology
- Cayman Chemical
- DC Chemicals
- Medical Isotopes, Inc.
- Sigma-Aldrich
- Tocris
- TRC
- Usbiological
Package
- 10
- 1mg
- 5mg
- 10mg
- 25mg
- 100MG
- 0.1g
- 250mg
- 1g
- Manufactureraablocks
- Product numberAA001MH3
- Product description2-Pyrrolidinecarboxamide,1-[[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-,(2S)- ≥98%
- Packaging5mg
- Price$222
- Updated2021-12-16
- Buy
- Manufactureraablocks
- Product numberAA001MH3
- Product description2-Pyrrolidinecarboxamide,1-[[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-,(2S)- ≥98%
- Packaging10mg
- Price$368
- Updated2021-12-16
- Buy
- Manufactureraablocks
- Product numberAA001MH3
- Product description2-Pyrrolidinecarboxamide,1-[[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-,(2S)- ≥98%
- Packaging25mg
- Price$720
- Updated2021-12-16
- Buy
- ManufacturerACHEMBLOCK
- Product numberH-8660
- Product description(2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide 98%
- Packaging5MG
- Price$245
- Updated2021-12-16
- Buy
- ManufacturerACHEMBLOCK
- Product numberH-8660
- Product description(2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide 98%
- Packaging100MG
- Price$1950
- Updated2021-12-16
- Buy
- ManufacturerAHH
- Product numberMT-04948
- Product description(2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide 98%
- Packaging0.1g
- Price$465
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product numberSYN5553
- Product descriptionRelcovaptan
- Packaging10mg
- Price$273
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0004734
- Product description(2S)-1-[[(2R,3S)-5-CHLORO-3-(2-CHLOROPHENYL)-1-[(3,4-DIMETHOXYPHENYL)SULFONYL]-2,3-DIHYDRO-3-HYDROXY-1H-INDOL-2-YL]CARBONYL]-2-PYRROLIDINECARBOXAMIDE 95.00%
- Packaging5MG
- Price$303.6
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0004734
- Product description(2S)-1-[[(2R,3S)-5-CHLORO-3-(2-CHLOROPHENYL)-1-[(3,4-DIMETHOXYPHENYL)SULFONYL]-2,3-DIHYDRO-3-HYDROXY-1H-INDOL-2-YL]CARBONYL]-2-PYRROLIDINECARBOXAMIDE 95.00%
- Packaging10MG
- Price$842.87
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB7013
- Product descriptionSR 49059
- Packaging10mg
- Price$353
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number17972
- Product descriptionSR 49059 ≥98%
- Packaging1mg
- Price$49
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number17972
- Product descriptionSR 49059 ≥98%
- Packaging5mg
- Price$168
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number17972
- Product descriptionSR 49059 ≥98%
- Packaging10mg
- Price$310
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number17972
- Product descriptionSR 49059 ≥98%
- Packaging25mg
- Price$651
- Updated2024-03-01
- Buy
- ManufacturerDC Chemicals
- Product numberDC8603
- Product descriptionSR 49059 >98%
- Packaging100mg
- Price$850
- Updated2021-12-16
- Buy
- ManufacturerDC Chemicals
- Product numberDC8603
- Product descriptionSR 49059 >98%
- Packaging250mg
- Price$1600
- Updated2021-12-16
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
aablocks | AA001MH3 | 2-Pyrrolidinecarboxamide,1-[[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-,(2S)- ≥98% | 5mg | $222 | 2021-12-16 | Buy |
aablocks | AA001MH3 | 2-Pyrrolidinecarboxamide,1-[[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-,(2S)- ≥98% | 10mg | $368 | 2021-12-16 | Buy |
aablocks | AA001MH3 | 2-Pyrrolidinecarboxamide,1-[[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-,(2S)- ≥98% | 25mg | $720 | 2021-12-16 | Buy |
ACHEMBLOCK | H-8660 | (2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide 98% | 5MG | $245 | 2021-12-16 | Buy |
ACHEMBLOCK | H-8660 | (2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide 98% | 100MG | $1950 | 2021-12-16 | Buy |
AHH | MT-04948 | (2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide 98% | 0.1g | $465 | 2021-12-16 | Buy |
AK Scientific | SYN5553 | Relcovaptan | 10mg | $273 | 2021-12-16 | Buy |
American Custom Chemicals Corporation | API0004734 | (2S)-1-[[(2R,3S)-5-CHLORO-3-(2-CHLOROPHENYL)-1-[(3,4-DIMETHOXYPHENYL)SULFONYL]-2,3-DIHYDRO-3-HYDROXY-1H-INDOL-2-YL]CARBONYL]-2-PYRROLIDINECARBOXAMIDE 95.00% | 5MG | $303.6 | 2021-12-16 | Buy |
American Custom Chemicals Corporation | API0004734 | (2S)-1-[[(2R,3S)-5-CHLORO-3-(2-CHLOROPHENYL)-1-[(3,4-DIMETHOXYPHENYL)SULFONYL]-2,3-DIHYDRO-3-HYDROXY-1H-INDOL-2-YL]CARBONYL]-2-PYRROLIDINECARBOXAMIDE 95.00% | 10MG | $842.87 | 2021-12-16 | Buy |
ApexBio Technology | B7013 | SR 49059 | 10mg | $353 | 2021-12-16 | Buy |
Cayman Chemical | 17972 | SR 49059 ≥98% | 1mg | $49 | 2024-03-01 | Buy |
Cayman Chemical | 17972 | SR 49059 ≥98% | 5mg | $168 | 2024-03-01 | Buy |
Cayman Chemical | 17972 | SR 49059 ≥98% | 10mg | $310 | 2024-03-01 | Buy |
Cayman Chemical | 17972 | SR 49059 ≥98% | 25mg | $651 | 2024-03-01 | Buy |
DC Chemicals | DC8603 | SR 49059 >98% | 100mg | $850 | 2021-12-16 | Buy |
DC Chemicals | DC8603 | SR 49059 >98% | 250mg | $1600 | 2021-12-16 | Buy |
Properties
Melting point :158-160oC
Boiling point :868.0±75.0 °C(Predicted)
Density :1.499±0.06 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: ≥10mg/mL
form :powder
pka :10.95±0.40(Predicted)
color :white to off-white
optical activity :[α]/D -180 to -190°, c = 0.3 in chloroform-d
Stability :Hygroscopic
Boiling point :868.0±75.0 °C(Predicted)
Density :1.499±0.06 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: ≥10mg/mL
form :powder
pka :10.95±0.40(Predicted)
color :white to off-white
optical activity :[α]/D -180 to -190°, c = 0.3 in chloroform-d
Stability :Hygroscopic
Safety Information
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Signal word: | Warning | |||||||||||||||||||||
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Description
SR 49059 is a selective, nonpeptide antagonist of the V1a subtype of the vasopressin receptor (Ki = 1.1-6.3 nM in human). It demonstrates ≥2 orders of magnitude lower affinity for V1b, V2, and oxytocin receptors and does not exhibit any intrinsic agonist activity. SR 49059 can inhibit arginine vasopressin-induced human platelet aggregation with an IC50 value of 3.7 nM.More related product prices
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