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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
6-chloro-2,3-dihydro-1H-quinolin-4-one 6-氯-2,3-二氢喹啉-4-酮 21617-20-9 详细
2,3-dihydro-1-benzofuran-5-amine 2,3-二氢-1-苯并呋喃-5-胺 42933-43-7 详细
6-bromocinnoline 6-溴曾嗪 318276-72-1 详细
benzyl 2,4-dichloro-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-7-carboxylate 苯甲基 2,4-二氯-5H,6H,7H,8H,9H-嘧啶并[4,5-d]氮杂卓-7-甲酸基酯 1207362-38-6 详细
(1S)-indan-1-amine;hydrochloride (S)-1-氨基茚满盐酸盐 32457-23-1 详细
tert-butyl 4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxylate 叔-丁基 4-氧亚基-3H,4H,5H,6H,7H-吡咯并[3,4-d]嘧啶-6-甲酸基酯 1229455-14-4 详细
tert-butyl 6-amino-2-oxo-1,2,3,4-tetrahydroquinoline-1-carboxylate 叔-丁基 6-氨基-2-氧亚基-1,2,3,4-四氢喹啉-1-甲酸基酯 1788054-94-3 详细
7-(difluoromethyl)-1,2,3,4-tetrahydroquinoline 7-(二氟甲基)-1,2,3,4-四氢喹啉 1783624-20-3 详细
6-bromo-2,2-dimethyl-3,4-dihydro-1H-quinoline 6-溴-2,2-二甲基-1,2,3,4-四氢喹啉 199186-78-2 详细
7-bromo-5-methyl-1,2,3,4-tetrahydroisoquinoline 7-bromo-5-methyl-1,2,3,4-tetrahydroisoquinoline 1934800-64-2 详细
ethyl 3-chloro-5H,6H,7H,8H-pyrido[4,3-c]pyridazine-6-carboxylate 6-N-CARBETHOXY-3-CHLORO-7,8-DIHYDRO-5H-PYRIDO[4,3-C]PYRIDAZINE 39715-99-6 详细
methyl 3-methylindoline-4-carboxylate;hydrochloride 甲基 3-甲基-2,3-二氢-1H-吲哚-4-羧酸盐酸盐 2387595-76-6 详细
3,4-dihydro-2H-1,4-benzoxazine-7-carboxylic acid 3,4-二氢-2H-1,4-苯并噁嗪-7-羧酸 851202-96-5 详细
5-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid 5-乙基-4,5,6,7-四氢-2H-吲唑-3-羧酸 856437-81-5 详细
6-chloro-1H,2H,3H-pyrrolo[3,2-c]pyridine 6-氯-2,3-二氢-5-氮杂吲哚 23596-25-0 详细
tert-butyl 7,8-dihydro-5H-pyrido[4,3-d]pyrimidine-6-carboxylate 7,8-二氢吡啶并[4,3-D]嘧啶-6(5H)-甲酸叔丁酯 192869-49-1 详细
2-chloro-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole 2-CHLORO-5H,6H,7H-PYRROLO[1,2-A]IMIDAZOLE 91417-91-3 详细
4-hydroxy-1,2,5,6,7,8-hexahydroquinolin-2-one 4-羟基-1,2,5,6,7,8-六氢喹啉-2-酮 56517-59-0 详细
7-bromo-4-chloro-indan-1-one 149965-64-0 149965-64-0 详细
6-chloro-5-nitro-indoline 6-氯-5-硝基-二氢吲哚 172078-32-9 详细
5,6,7,8-tetrahydroquinolin-5-amine 5,6,7,8-四氢喹啉-5-胺 71569-15-8 详细
methyl 1,2,3,4-tetrahydroisoquinoline-5-carboxylate hydrochloride 甲基 1,2,3,4-四氢异喹啉-5-甲酸基酯盐酸 1035700-06-1 详细
7-bromo-2H-phthalazin-1-one 二氮杂萘-1(2H)-酮 152265-57-1 详细
isoindolin-4-amine;dihydrochloride 4-氨基异吲哚林盐酸盐 92259-85-3 详细
O5-tert-butyl O2-ethyl 6,7-dihydro-4H-thiazolo[5,4-c]pyridine-2,5-dicarboxylate 5-BOC-4,5,6,7-四氢-1,3-噻唑并[5,4-C]吡啶-2-甲酸乙酯 1053656-51-1 详细
tert-butyl 8-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxylate TERT-BUTYL 8-(4,4,5,5-TETRAMETHYL-1,3,2-DIOXABOROLAN-2-YL)-3,4-DIHYDROISOQUINOLINE-2(1H)-CARBOXYLATE 893566-73-9 详细
2-tert-butyl 7-methyl 1,2,3,4-tetrahydroisoquinoline-2,7-dicarboxylate 2-叔-丁基 7-甲基 1,2,3,4-四氢异喹啉-2,7-二甲酸基酯 960305-54-8 详细
2-(4-oxo-3,4-dihydrophthalazin-1-yl)acetic acid 2-(4-氧亚基-3,4-二氢酞嗪-1-基)乙酸 25947-11-9 详细
1,2,3,4-tetrahydro-1,8-naphthyridin-2-one 1,2,3,4-四氢-1,8-萘啶-2-酮 40000-79-1 详细
1,2,3,4-tetrahydroisoquinoline-7-carbonitrile 1,2,3,4-四氢异喹啉-7-甲腈 149355-52-2 详细
5-tert-butoxycarbonyl-7-methyl-2,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-3-carboxylic acid 5-叔丁氧基羰基-7-甲基-2,4,6,7-四氢吡唑[4,3-C]吡啶-3-羧酸 2171296-03-8 详细
6-bromo-1H-cinnolin-4-one 6-溴-4(1H)-噌啉酮 552330-87-7 详细
6-tert-butyl 3-ethyl 2-amino-4H,5H,6H,7H-thieno[2,3-c]pyridine-3,6-dicarboxylate 6-叔-丁基 3-乙基 2-氨基-4H,5H,6H,7H-噻吩并[2,3-c]吡啶-3,6-二甲酸基酯 193537-14-3 详细
tert-butyl 2-amino-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxylate 2-氨基-5H-吡咯并[3,4-D]嘧啶-6(7H)-甲酸叔丁酯 1105187-42-5 详细
methyl 2-[(3S)-6-hydroxy-2,3-dihydro-1-benzofuran-3-yl]acetate 甲基 2-[(3S)-6-羟基-2,3-二氢-1-苯并呋喃-3-基]醋酸盐 1000414-38-9 详细
5-tert-butyl 3-ethyl 2-amino-4H,5H,6H,7H-thieno[3,2-c]pyridine-3,5-dicarboxylate 5-叔-丁基 3-乙基 2-氨基-4H,5H,6H,7H-噻吩并[3,2-c]吡啶-3,5-二甲酸基酯 1101856-88-5 详细
1,2,3,4-tetrahydroisoquinolin-7-ylmethanol;hydrochloride (1,2,3,4-tetrahydroisoquinolin-7-yl)methanol hydrochloride 2152636-99-0 详细
4-chloro-2,3-dihydro-1H-pyrrolo[3,4-c]pyridine;hydrochloride 4-氯-2,3-二氢-1H-吡咯并[3,4-C]吡啶盐酸盐 2387597-05-7 详细
3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6,7-dihydro-4H-pyrazolo[5,1-c][1,4]oxazine 6,7-二氢-4H-吡唑并[5,1-C][1,4]噁嗪-3-硼酸频哪醇酯 2057507-08-9 详细
ethyl 4-oxo-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate 乙基 4-氧亚基-4H,5H,6H,7H-吡唑并[1,5-a]吡嗪-2-甲酸基酯 951626-95-2 详细
methyl 3,4-dihydro-2H-1,4-benzoxazine-7-carboxylate 3,4-二氢-2H-苯并[1,4]恶嗪-7-甲酸甲酯 142166-01-6 详细
(2,3-dihydro-1-benzofuran-6-yl)methanamine 6-COUMARANMETHYLAMINE 55746-20-8 详细
7-bromo-4-methoxy-indan-1-one 7-溴-4-甲氧基茚酮 959058-59-4 详细
5-chloro-2-methylsulfanyl-pyrido[4,3-d]pyrimidine 5-氯-2-(甲巯基)吡啶并[4,3-D]嘧啶 1255099-52-5 详细
2-[(tert-butoxy)carbonyl]-5,7-dichloro-1,2,3,4-tetrahydroisoquinoline-6-carboxylic acid 2-[(叔-丁氧基)羰基]-5,7-二氯-1,2,3,4-四氢异喹啉-6-羧酸 851784-82-2 详细
4-fluoro-2,3-dihydrofuro[2,3-b]pyridine 4-氟-2H,3H呋喃并[2,3-b]吡啶 1818847-50-5 详细
7-bromo-3-chloro-pyrido[2,3-b]pyrazine 7-溴-3-氯吡啶并[2,3-B]吡嗪 1240594-95-9 详细
4-fluoro-2,3-dihydro-1H-inden-1-one 4-氟-1-茚酮 699-99-0 详细
3-bromo-6H-pyrido[2,3-d]pyridazin-5-one 3-溴-6H-吡啶并[2,3-D]哒嗪-5-酮 1426245-35-3 详细
8-benzyl-2,4-dichloro-5,6,7,9-tetrahydropyrimido[4,5-c]azepine 2,4-二氯-6,7,8,9-四氢-8-(苯甲基)-5H-嘧啶[4,5-C]氮卓 2617829-46-4 详细
5-nitroindan-2-one 5-硝基-2-茚酮 116530-60-0 详细
7-bromo-1H-quinoxalin-2-one 7-溴-2(1H)-喹喔啉酮 82031-32-1 详细
7-bromo-3H,4H-pyrido[3,2-d]pyrimidin-4-one 7-溴-3H,4H-吡啶并[3,2-d]嘧啶-4-酮 573675-29-3 详细
4,6-dichloro-7-fluoro-1H,2H,3H-pyrrolo[3,4-c]pyridin-3-one 4,6-二氯-7-氟-1H-吡咯并[3,4-C]吡啶-3(2H)-酮 1312693-69-8 详细
7-bromo-4-nitro-indan-1-one 7-溴-4-硝基茚满-1-酮 1260018-07-2 详细
tert-butyl 3-iodo-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-5-carboxylate 5-BOC-3-碘-5,6,7,8-四氢-4H-吡唑并[1,5-A][1,4]二氮杂卓 1823263-02-0 详细
2-(6-hydroxy-2,3-dihydro-1-benzofuran-3-yl)acetic acid 2-(6-羟基-2,3-二氢-1-苯并呋喃-3-基)乙酸 1000414-37-8 详细
tert-butyl 3-amino-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate Tert-Butyl 3-Amino-6,7-Dihydropyrazolo[1,5-A]Pyrazine-5(4H)-Carboxylate(WX141188) 1391733-15-5 详细
3-fluoro-6,7-dihydrocyclopenta[b]pyridin-5-one 3-氟-6,7-二氢环戊二烯并[B]吡啶-5-酮 1196156-82-7 详细
N-(7-fluoro-8-methyl-4-oxo-tetralin-5-yl)acetamide N-(3-氟-4-甲基-8-氧代-5,6,7,8-四氢-1-萘基)乙酰胺 143655-58-7 详细
tert-butyl 6-bromo-4,4-difluoro-1,3-dihydroisoquinoline-2-carboxylate 2306276-51-5 详细
2-(trifluoromethyl)-6,7-dihydro-5H-cyclopenta[b]pyridin-5-amine;dihydrochloride 2-(三氟甲基)-6,7-二氢-5H-环戊[B]吡啶-5-胺二盐酸盐 2832389-56-5 详细
2,3,4,5-tetrahydro-1H-1,5-benzodiazepin-2-one 1,3,4,5-四氢-苯并[B][1,4]二氮杂革-2-酮 5755-07-7 详细
6-bromo-2-chloropyrido[2,3-d]pyrimidine 6-溴-2-氯吡啶并[2,3-d]嘧啶 1234616-65-9 详细
5H,6H,7H-pyrrolo[3,4-d]pyrimidine hydrochloride 6,7-二氢-5H-吡咯并[3,4-D]嘧啶盐酸 1187830-46-1 详细
2-methyl-6,7-dihydro-5H-indazol-4-one 2-甲基-6,7-二氢-2H-吲唑-4(5H)-酮 1027617-67-9 详细
1',4',6',7'-tetrahydrospiro[[1,3]dioxolane-2,5'-indazole 2',4',6',7'-四氢螺[1,3-二氧戊环-2,5'-吲唑 1204218-41-6 详细
6-bromo-1-methyl-1,2,3,4-tetrahydroquinolin-2-one 6-溴-1-甲基-1,2,3,4-四氢喹啉-2-酮 1092523-03-9 详细
6-[(tert-butoxy)carbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carboxylic acid 6-[(叔-丁氧基)羰基]-5,6,7,8-四氢-1,6-萘啶-3-羧酸 1341036-28-9 详细
6-chloropyrido[3,4-d]pyrimidin-4-amine 6-chloropyrido[3,4-d]pyrimidin-4-amine 1289187-97-8 详细
tert-butyl 3-iodo-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-5-carboxylate 3-碘-6,7-二氢吡唑并[1,5-A]吡嗪-5(4H)-羧酸叔丁酯 1823229-68-0 详细
(1S)-tetralin-1-amine (S)-1,2,3,4-四氢-1-萘胺 23357-52-0 详细
7-Amino-3,4-dihydro-2(1H)-quinolinone 7-氨基-3,4-二氢-1H-喹啉-2-酮 22246-07-7 详细
2,3,4,5-tetrahydro-1H-1-benzazepin-2-one 1,3,4,5-四氢-2H-1-苯并氮杂卓-2-酮 4424-80-0 详细
5,7-dichloro-3H-pyrido[4,3-d]pyrimidin-4-one 5,7-二氯吡啶并[4,3-D]嘧啶-4(3H)-酮 918898-11-0 详细
3-bromo-4H,5H,6H-pyrrolo[1,2-b]pyrazole 3-BROMO-5, 6-DIHYDRO-4H-PYRROLO[1, 2-B]PYRAZOLE 174790-35-3 详细
5,5-dimethyl-3-(tetramethyl-1,3,2-dioxaborolan-2-yl)-4H,5H,6H-pyrrolo[1,2-b]pyrazole 4H-Pyrrolo[1,2-b]pyrazole, 5,6-dihydro-5,5-dimethyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)- 2057507-59-0 详细
2-chloro-8-iodopyrido[4,3-d]pyrimidine 2-chloro-8-iodopyrido[4,3-d]pyrimidine 1562987-94-3 详细
7-(trifluoromethyl)-3,4-dihydro-1H-2-benzopyran-4-one 7-(三氟甲基)异色满-4-酮 1344725-51-4 详细
1-methylindoline 1-甲基吲哚啉 824-21-5 详细
5,6-dichloro-2,3-dihydrobenzofuran-3-amine;hydrochloride 5,6-二氯-2,3-二氢苯并呋喃-3-胺盐酸盐 2725790-82-7 详细
2,4-dichloro-5,6,7,8-tetrahydroquinazoline 2,4-二氯-6,7-二氢-5H-环戊并嘧啶 1127-85-1 详细
3,4-dihydro-2H-1-benzopyran-4-carboxylic acid 3,4-DIHYDRO-2H-1-BENZOPYRAN-4-CARBOXYLIC ACID 20426-80-6 详细
methyl tetralin-5-carboxylate 茚满-4-甲酸甲酯 66193-59-7 详细
3-bromo-5,6-dihydrocyclopenta[b]pyridin-7-one 3-溴-5H-2,3-环戊烯并吡啶-7(6H)-酮 1336955-89-5 详细
5-[(tert-butoxy)carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxylic acid 5-[(叔-丁氧基)羰基]-4H,5H,6H,7H-[1,2]噁唑并[4,5-c]吡啶-3-羧酸 912265-93-1 详细
3-bromo-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine hydrochloride 3-溴-4,5,6,7-四氢吡唑并[1,5-A]吡嗪盐酸盐 2059994-83-9 详细
7-bromo-4-(trifluoromethyl)indan-1-one 7-溴-4-(三氟甲基)茚满-1-酮 1337833-33-6 详细
7-amino-8-bromo-tetralin-1-one 1(2H)-Naphthalenone, 7-amino-8-bromo-3,4-dihydro- 214697-98-0 详细
ethyl 4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridine-2-carboxylate;hydrochloride 4,5,6,7-四氢-5-氮杂吲哚-2-甲酸乙酯盐酸盐 2504201-65-2 详细
5H,6H,7H,8H-imidazo[1,5-a]pyrazine dihydrochloride 5H,6H,7H,8H-咪唑并[1,5-a]吡嗪二盐酸 165894-10-0 详细
methyl 2-(4-oxo-3,4-dihydrophthalazin-1-yl)acetate METHYL3,4-DIHYDRO-4-OXO-1-PHTHALAZINEACETATE 25947-14-2 详细
7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine hydrochloride 7-甲氧基-2,3,4,5-四氢-1H-3-苯氮杂卓盐酸 17639-46-2 详细
4,7-dichloropyrido[3,2-d]pyrimidine N-甲基-3-氨基吡啶 917757-12-1 详细
5-tert-butoxycarbonyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid 5-N-BOC 4,5,6,7-四氢吡唑并[1,5-A]吡啶-2-羧酸 1209492-73-8 详细
1-tert-butyl 6-methyl 5-bromo-2,3-dihydro-1h-indole-1,6-dicarboxylate 1-叔-丁基 6-甲基 5-溴-2,3-二氢-1h-吲哚-1,6-二甲酸基酯 1788044-06-3 详细
8-chloro-2-(methylsulfanyl)pyrido[3,4-d]pyrimidine 8-氯-2-(甲基巯基)吡啶并[3,4-d]嘧啶 1578245-95-0 详细
5-chloro-6-nitro-indoline 5-氯-6-硝基-二氢吲哚 2007919-15-3 详细
4-bromo-7-fluoro-indane 4-溴-7-氟-2,3-二氢-1H-茚 2332943-95-8 详细
7-bromo-2,3-dihydropyrazolo[5,1-b]oxazole 7-溴-2,3-二氢吡唑并[5,1-B]恶唑 1554086-90-6 详细
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