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  •       科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。 科学驱动的设计策略确保分子砌块的新颖性和多样性,提高苗头化合物和先导化合物的筛选和优化效率; 针对特定化学系列不断积累化学知识和经验,快速交付具有挑战性的化合物; 完备的合成、工艺开发和生产能力,以及稳定的原料供应管理,可持续供应从克级、公斤级到吨级的分子砌块产品,支持新药研发、开发至商业化需求。
英文名称 中文名称 CAS号 操作
Canertinib 卡奈替尼 267243-28-7 详细
1,7-naphthyridine-2-carboxylic acid 1,7-萘啶-2-羧酸 316155-87-0 详细
(2S)-2-[[(2S)-2-amino-3-phenyl-propanoyl]amino]-3-(1H-indol-3-yl)propanoic acid H-PHE-TRP-OH 24587-41-5 详细
6-chlorotetralin-1-one 6-氯-3,4-二氢-2H-1-萘酮 26673-31-4 详细
8-ethyl-7-fluoro-3-(methoxymethoxy)naphthalen-1-ol 8-乙基-7-氟-3-(甲氧基甲氧基)萘-1-醇 2621932-46-3 详细
3-cyclopropyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4-(trifluoromethyl)aniline 3-环丙基-5-(4,4,5,5-四甲基-1,3,2-二噁硼戊环-2-基)-4-(三氟甲基)苯胺 2820116-37-6 详细
N-[4-[(2R)-1-(4-acetamido-2-fluoro-phenyl)pyrrolidin-2-yl]thiazol-2-yl]-1-[(2-fluoro-4-pyridyl)methyl]pyrrole-2-carboxamide 2763270-65-9 详细
5-bromo-2,4-difluorobenzene-1-sulfonyl chloride 5-溴-2,4-二氟苯磺酰氯 287172-61-6 详细
INH-1 N-[4-(2,4-二甲基苯基)-2-噻唑基]苯甲酰胺 313553-47-8 详细
(1S,2S)-1,2-diphenylethane-1,2-diamine (1S,2S)-1,2-二苯基乙烷-1,2-二胺 29841-69-8 详细
7-bromo-2,4-dichloro-6-methoxy-pyrido[3,2-d]pyrimidine 7-溴-2,4-二氯-6-甲氧基嘧啶[3,2-D]嘧啶 2577287-84-2 详细
5-(3-fluorophenyl)oxazole Oxazole, 5-(3-fluorophenyl)- (9CI) 243455-58-5 详细
tert-butyl 2-(trifluoromethylsulfonyloxy)spiro[5,6-dihydropyrrolo[1,2-b]pyrazole-4,3'-pyrrolidine]-1'-carboxylate 2'-(((三氟甲基)磺酰基)氧基)-5',6'-二氢螺[吡咯烷-3,4'-吡咯并[1,2-B]吡唑]-1-羧酸叔丁酯 2640496-81-5 详细
(2S,4R)-1-[(2S)-2-[5-[[2-[2,3-difluoro-6-(2-morpholinothiazol-4-yl)phenoxy]acetyl]amino]pentanoylamino]-3,3-dimethyl-butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methylthiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide 2488296-74-6 详细
8-bromo-2-ethylsulfanyl-6-methyl-chromen-4-one 8-溴-2-(乙硫基)-6-甲基-4H-色烯-4-酮 2715284-54-9 详细
2-chloro-5,6-dihydro-4H-1,3-benzothiazol-7-one 2-氯-5,6-二氢苯并[D]噻唑-7(4H)-酮 330203-55-9 详细
tert-butyl 4-[2-(hydroxymethyl)phenyl]piperidine-1-carboxylate 255051-62-8 255051-62-8 详细
7-bromo-4H-1,4-benzoxazin-3-one 7-溴-2H-1,4-苯并嗪-3(4H)-酮 321436-06-0 详细
Harringtonin 三尖杉酯碱 26833-85-2 详细
6-bromo-8-methyl-3,4-dihydro-2H-isoquinolin-1-one 6-溴-8-甲基-3,4-二氢异喹啉-1(2H)-酮 2426763-19-9 详细
1-bromo-5-fluoro-naphthalene 1-溴-5-氟萘 315-56-0 详细
3-fluoro-6,7-dihydro-5H-pyrrolo[3,4-b]pyridine;dihydrochloride 3-氟-6,7-二氢-5H-吡咯并[3,4-B]吡啶二盐酸盐 2613381-76-1 详细
2-amino-1-(3-hydroxy-2,6-dimethyl-phenyl)-5,6-dimethyl-pyrrolo[2,3-b]pyridine-3-carboxamide RP-6306 2719793-90-3 详细
1,1-dioxo-3,5-dihydro-2H-4,1benzoxathiepine-8-carboxylic acid 2,3-二氢-5H-4,1-苯并氧硫杂卓-8-羧酸1,1-二氧化物 2771132-16-0 详细
2-chloro-6-(1-methylpyrazol-4-yl)pyrimidine-4-carboxylic acid 2839856-36-7 详细
2-bromo-5,5-difluoro-4,6-dihydropyrrolo[1,2-b]pyrazole 2711994-99-7 详细
BAY-41-8543 BAY-41-8543 256498-66-5 详细
(1R,2S,5S)-N-[(1S)-1-cyano-2-[(3S)-2-oxopyrrolidin-3-yl]ethyl]-3-[(2S)-3,3-dimethyl-2-[(2,2,2-trifluoroacetyl)amino]butanoyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxamide 帕罗韦德 2628280-40-8 详细
Cediranib 西地尼布 288383-20-0 详细
8'-fluoro-7'-iodo-6'-(2-methoxyethoxymethoxy)spiro[1,3-dioxolane-2,2'-tetralin 8'-氟代-7'-碘代-6'-((2-甲氧基乙氧基)甲氧基)-3',4'-二氢-1'H-螺环[[1,3]二氧戊环-2,2'-萘] 2489407-90-9 详细
2,4,7-trichloro-8-fluoro-1,6-naphthyridine-3-carbonitrile 2,4,7-三氯-8-氟-1,6-萘啶-3-腈 2769863-96-7 详细
(3R,5S)-3-methyl-5-[4-(trifluoromethyl)phenyl]morpholine 2655519-30-3 详细
(7S)-2-bromo-7-methyl-5,6-dihydropyrrolo[1,2-a]imidazol-7-ol 2639837-09-3 详细
2,4,6,8-tetrachloropyrimido[5,4-d]pyrimidine 四氯嘧啶并[5,4-D]嘧啶 32980-71-5 详细
1-(diethoxyphosphorylmethyl)-4-nitro-benzene 二乙基(4-硝基苯甲基)磷酸盐 2609-49-6 详细
7-fluoronaphthalen-1-ol 7-氟萘-1-醇 3132-92-1 详细
tert-butyl 7-acetyl-1,2,4,5-tetrahydro-3-benzazepine-3-carboxylate 264264-31-5 详细
1,2,3,4-tetrahydroquinolin-6-ol 6-羟基-1,2,3,4-四氢喹啉 3373-00-0 详细
(4R)-2-amino-4-ethynyl-4-methyl-6,7-dihydro-5H-benzothiophene-3-carbonitrile (R)-2-氨基-4-乙炔基-4-甲基-4,5,6,7-四氢苯并[B]噻吩-3-甲腈 2749965-89-5 详细
7-methoxychromane-3-carboxylic acid 7-甲氧基苯并四氢吡喃-3-甲酸 3187-51-7 详细
SB-431542 SB-431542 301836-41-9 详细
2,4,7,8-tetrachloropyrido[4,3-d]pyrimidine 2,4,7,8-四氯吡啶并[4,3-D]嘧啶 2454396-63-3 详细
5-chlorotetralin-1-one 5-氯-Α-四氢萘酮 26673-30-3 详细
5,6,7,8-tetrahydro-1,7-naphthyridin-8-one 6,7-二氢-1,7-萘啶-8(5H)-酮 301666-63-7 详细
4-(trifluoromethoxy)benzoic acid 4-三氟甲氧基苯甲酸 330-12-1 详细
7-fluorotetralin-1-one 7-氟-Α-四氢萘酮 2840-44-0 详细
2-(5-fluoro-2-methyl-1H-inden-3-yl)acetic acid (5-氟-2-甲基-1H-茚-3-基)乙酸 32004-66-3 详细
tert-butyl (2S)-2-(cyanomethyl)-4-(2,7-dichloro-8-fluoro-pyrido[4,3-d]pyrimidin-4-yl)piperazine-1-carboxylate 2454396-81-5 详细
7-(bromomethyl)-8-fluoro-3-methyl-1H-quinoxalin-2-one 7-(溴甲基)-8-氟-3-甲基喹喔啉-2(1H)-酮 2756333-93-2 详细
2-bromo-6-methyl-6,7-dihydro-5H-pyrazolo[1,5-a]pyrazin-4-one 2468022-90-2 详细
(3S)-3-(5-bromo-1-oxo-isoindolin-2-yl)piperidine-2,6-dione (3S)-3-(5-溴-1-氧代-异吲哚啉-2-基)哌啶-2,6-二酮 2829898-76-0 详细
4-(5-chloro-2-methoxy-phenyl)-6-methyl-pyridine-3-carboxylic acid 4-(5-氯-2-甲氧基苯基)-6-甲基烟酸 2782813-27-6 详细
(7R)-2-bromo-7-methyl-5,6-dihydropyrrolo[1,2-a]imidazol-7-ol 2639837-10-6 详细
tert-butyl 2-oxospiro[indoline-3,4-piperidine]-1-carboxylate 1'-BOC-1,2-二氢-2-氧代-螺[3H-吲哚-3,4'-哌啶] 252882-60-3 详细
3-(Diphenylphosphino)propionic Acid 3-(二苯基膦)丙酸 2848-01-3 详细
6,7-dichlorotetralin-1-one 6,7-二氯-3,4-二氢-1H-2-萘酮 25095-57-2 详细
tert-butyl N-[2-(3-hydroxy-4-methoxy-phenyl)ethyl]carbamate (3-羟基-4-甲氧基苯乙基)氨基甲酸叔丁酯 31493-49-9 详细
methyl 3-bromo-5-fluoro-benzoate 3-溴-5-氟苯甲酸甲酯 334792-52-8 详细
2-hydroxy-4-nitro-benzaldehyde 2-羟基-4-硝基苯甲醛 2460-58-4 详细
1-bromo-8-chloro-3-(methoxymethoxy)naphthalene 1-溴-8-氯-3-(甲氧基甲氧基)萘 2454490-96-9 详细
2-(7,8-difluoro-1-naphthyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(7,8-二氟萘-1-基)-4,4,5,5-四甲基-1,3,2-二氧硼烷 2454490-85-6 详细
pelitinib 培利替尼 257933-82-7 详细
3-chloro-4-(1-methylbenzimidazol-5-yl)oxy-aniline 2682003-53-6 详细
methyl (1R,3R,4R,5S)-3-[(2R,3R,4R,5R,6R)-3-(allyloxycarbonylamino)-4,5-dihydroxy-6-(hydroxymethyl)tetrahydropyran-2-yl]oxy-5-ethyl-4-[(2S,3S,4R,5R,6S)-3,4,5-tribenzyloxy-6-methyl-tetrahydropyran-2-yl]oxy-cyclohexanecarboxylate (1R,3R,4R,5S)-3-[[(2R,3R,4R,5R,6R)-3-[[(烯丙基氧基)羰基]氨基]-4,5-二羟基-6-(羟甲基)四氢-2H-吡喃-2-基]氧基]-5-乙基-4-[[(2S,3S,4R,5R,6S)-3,4,5-三(苄氧基)-6-甲基四氢-2H-吡喃-2-基]氧基]环己烷甲酸甲酯 2609644-29-1 详细
2,5,7-trichloro-8-fluoro-3H-pyrido[4,3-d]pyrimidin-4-one 叔丁基(1R,4R,6S)-6-(羟甲基)-2,5-二氮杂二环[2.2.1]庚烷-2-羧酸盐 2836267-81-1 详细
(21R)-5-cyano-4-fluoro-9,9-dioxo-16-oxa-9λ-thia-1,8-diazatetracyclo[19.4.0.02,.01,1]pentacosa-2,4,6,10,12,14-hexaene-12-carboxylic acid 2766037-03-8 详细
tert-butyl 4-oxo-7,9-dihydro-6H-pyrazino[1,2-a]pyrimidine-8-carboxylate 叔-丁基 4-羰基-7,9-二氢-6H-吡喃联氮基[1,2-A]嘧啶-8-羧酸酯 2828020-77-3 详细
N-[4-[(2R)-1-(4-acetamido-2,6-difluoro-phenyl)pyrrolidin-2-yl]thiazol-2-yl]-1-[(2-fluoro-4-pyridyl)methyl]pyrrole-2-carboxamide 2763270-63-7 详细
(2S,3S)-2,3-bis[(4-methylbenzoyl)oxy]butanedioic acid D-(+)-二对甲基苯甲酰酒石酸 32634-68-7 详细
1-methyl-4,5,6,7-tetrahydroindazole-3-carboxylic acid 1-甲基-4,5,6,7-四氢-1H-吲唑-3-羧酸 32286-99-0 详细
6-chloro-1,2,3,4-tetrahydroisoquinoline;hydrochloride 6-氯-1,2,3,4-四氢异喹啉盐酸盐 33537-97-2 详细
2-(oxiran-2-yl)acetic acid 2-(噁丙环-2-基)乙酸 33278-09-0 详细
Uracil arabinoside 阿糖尿苷 3083-77-0 详细
spiro[indene-1,4'-piperidine 螺[茚-1,4'-哌啶] 33042-66-9 详细
triisopropyl-[2-[6-(methoxymethoxy)-8-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-naphthyl]ethynyl]silane 三异丙基((6-(甲氧基甲氧基)-8-(4,4,5,5-四甲基-1,3,2-二氧杂硼硼烷-2-基)萘-1-基)乙炔基)硅烷 2621932-42-9 详细
7-(chloromethyl)-3-ethyl-1H-1,5-naphthyridin-2-one 7-(氯甲基)-3-乙基-1,5-萘啶-2(1H)-酮 2589531-78-0 详细
methyl 2-(5-hydroxy-1-methyl-pyrazol-4-yl)-6-methyl-pyridine-4-carboxylate 2573870-42-3 详细
2-[[rel-(1R,5S,6r)-3-azabicyclo[3.1.0]hexan-6-yl]methylsulfanyl]-1,3-benzothiazole;hydrochloride 2691954-45-5 详细
6-[[2-chloro-4-(trifluoromethyl)phenoxy]methyl]-4-ethyl-pyridine-2-carboxylic acid 化合物 MRGPRX4 MODULATOR-1 2492596-61-7 详细
4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxylic acid 吡唑[1,5-A] 4,5,6,7-四氢吡啶-3-羧酸 307307-97-7 详细
isopropyl N-[4-[(2R)-2-[2-[[1-[(2-fluoro-4-pyridyl)methyl]pyrrole-2-carbonyl]amino]thiazol-4-yl]pyrrolidin-1-yl]phenyl]carbamate 2763271-13-0 详细
spongosine GL101375 24723-77-1 详细
(2-chloro-4-(trifluoromethoxy)phenyl)boronic acid 2-氯-4-三氟甲氧基苯硼酸 345226-20-2 详细
3-oxo-2,3-dihydro-1H-indene-1-carboxylic acid 3-羰基-1-茚酸 29427-69-8 详细
2-(oxolan-3-yl)cyclohexan-1-one 2-(tetrahydrofuran-3-yl)cyclohexanone 31891-67-5 详细
3-(butylamino)-4-phenoxy-5-sulfamoylbenzoic acid 布美他尼 28395-03-1 详细
1-(bromomethyl)-4-phenyl-benzene 4-溴甲基联苯 2567-29-5 详细
BAY-41-2272 BAY 41-2272 256376-24-6 详细
8-ethyl-3-(methoxymethoxy)naphthalen-1-ol 8-乙基-3-(甲氧基甲氧基)萘-1-醇 2621932-58-7 详细
2-[8-ethyl-3-(methoxymethoxy)-1-naphthyl]-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(8-乙基-3-(甲氧基甲氧基)萘-1-基)-4,4,5,5-四甲基-1,3,2-二氧杂硼烷 2621932-60-1 详细
trans-4-[[(6-bromo-1,3-benzothiazol-2-yl)amino]methyl]cyclohexanecarboxylic acid 2664977-37-9 详细
4-methoxy-6-(pyrazol-1-ylmethyl)-1,2-benzoxazol-3-amine 6-((1H-吡唑-1-基)甲基)-4-甲氧基苯并[D]异噁唑-3-胺 2568912-43-4 详细
methyl 5,6,7,8-tetrahydro-1,7-naphthyridine-3-carboxylate;dihydrochloride 5,6,7,8-四氢-1,7-萘啶-3-羧酸甲酯二盐酸盐 2551116-71-1 详细
tert-butyl 4-(azetidin-3-ylmethyl)piperidine-1-carboxylate;hydrochloride 1-BOC-4-(氮杂环丁烷-3-基甲基)哌啶盐酸盐 2580216-69-7 详细
2-chloro-6-tetrahydrofuran-2-yl-pyrimidine-4-carboxylic acid 2737686-55-2 详细
7-(chloromethyl)-3-ethyl-1H-1,5-naphthyridin-2-one;hydrochloride 3-乙基-7-(氯甲基)-1,5-萘啶-2(1H)-酮盐酸盐 2589531-79-1 详细
6-bromo-1',1'-difluoro-spiro[2,3-dihydroisoquinoline-4,2'-cyclopropane]-1-one 2771025-18-2 详细
benzyl N-[2-tert-butyl-5-[trans-3-hydroxycyclopentyl]pyrazol-3-yl]carbamate REL-苄基(1-(叔丁基)-3-((1S,3S)-3-羟基环戊基)-1H-吡唑-5-基)氨基甲酸酯 2460255-79-0 详细
7-(bromomethyl)-3-ethyl-8-fluoro-1H-quinoxalin-2-one 7-(溴甲基)-3-乙基-8-氟-1H-喹喔啉-2-酮 2756334-33-3 详细
ethyl N-[4-[(2R)-2-[2-[[1-[(2-fluoro-4-pyridyl)methyl]pyrrole-2-carbonyl]amino]thiazol-4-yl]pyrrolidin-1-yl]phenyl]carbamate 噻唑杂质7 2763271-12-9 详细
产品总数:7268 产品页码:
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