| Identification | Back Directory | [Name]
Benzamide, 2-chloro-4-ethoxy-N-[[[6-[(1-methyl-4-piperidinyl)sulfonyl]-2-benzothiazolyl]amino]carbonyl]-5-(1H-pyrazol-1-yl)- | [CAS]
1143024-28-5 | [Synonyms]
GPR81 agonist 2
Benzamide, 2-chloro-4-ethoxy-N-[[[6-[(1-methyl-4-piperidinyl)sulfonyl]-2-benzothiazolyl]amino]carbonyl]-5-(1H-pyrazol-1-yl)- | [Molecular Formula]
C26H27ClN6O5S2 | [MOL File]
1143024-28-5.mol | [Molecular Weight]
603.11 |
| Hazard Information | Back Directory | [Uses]
GPR81 agonist 2 (compound 1) is a potent GPR81 agonist with EC50 values of 0.023, 0.123 μM for hGPR81, hGPR109A, respectively[1]. | [References]
[1] Davidsson ?, et al. Identification of novel GPR81 agonist lead series for target biology evaluation. Bioorg Med Chem Lett. 2020 Feb 15;30(4):126953. DOI:10.1016/j.bmcl.2020.126953 |
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Biorbyt Ltd.
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www.biorbyt.com |
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