| Identification | Back Directory | [Name]
(E)-(+/-)-2-AMINO-4-METHYL-5-PHOSPHONO-3-PENTENOIC ACID ETHYL ESTER | [CAS]
127910-32-1 | [Synonyms]
CGP 39551
2-Amino-4-methyl-5-phosphono-3 pentenoic acid carboxyethyl ester
(E)-(4-Amino-5-ethoxy-2-methyl-5-oxopent-2-en-1-yl)phosphonic acid
(E)-(+/-)-2-AMINO-4-METHYL-5-PHOSPHONO-3-PENTENOIC ACID ETHYL ESTER
(E)-(+/-)-2-AMINO-4-METHYL-5-PHOSPHONO-3-PENTENOIC ACID ETHYLESTHER
3-Pentenoic acid, 2-amino-4-methyl-5-phosphono-, 1-ethyl ester, (3E)-
3-Pentenoic acid, 2-amino-4-methyl-5-phosphono-, 1-ethyl ester, (E)-(+-)- | [Molecular Formula]
C8H16NO5P | [MDL Number]
MFCD00882474 | [MOL File]
127910-32-1.mol | [Molecular Weight]
237.19 |
| Chemical Properties | Back Directory | [Boiling point ]
434.1±55.0 °C(Predicted) | [density ]
1.312±0.06 g/cm3(Predicted) | [storage temp. ]
Desiccate at +4°C | [solubility ]
H2O: soluble15mg/mL, clear | [form ]
powder | [pka]
2.30±0.10(Predicted) | [color ]
white to beige | [Water Solubility ]
Soluble to 100 mM in water |
| Hazard Information | Back Directory | [Uses]
CGP 39551 is a potent, selective and competitive NMDA antagonist. | [Biological Activity]
Potent, selective and competitive NMDA antagonist (K i = 310 nM for inhibition of [ 3 H]-CPP binding in rat brain). Centrally active upon oral administration in vivo . | [in vivo]
CGP 39551 exhibits maximal electroshock-induced seizures in mice with the ED50 of 4 mg/kg (p.o.)[2].
Following chronic neonatal treatment with CGP 39551, adult rats show increased behavioral responses to the D2 dopamine receptor stimulation[3]. | [storage]
Desiccate at +4°C |
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