| Identification | Back Directory | [Name]
TRV-130 | [CAS]
1401031-39-7 | [Synonyms]
TRV130 HCl
Oliceridine HCl
TRV130 (hydrochloride)
TRV130 HCl (Oliceridine)
Oliceridine hydrochloride
Oliceridine HCl (TRV-130)
TRV-130 Hydrochloric Acid Salt
TRV130; TRV 130; TRV130; OLICERIDINE; OLICERIDINE HCL; OLICERIDINE HYDROCHLORIDE
TRV-130;TRV 130;TRV-130 HYDROCHLORIDE;TRV 130 HYDROCHLORIDE;OLICERIDINE HYDROCHLORIDE
(R)-N-((3-Methoxythiophen-2-yl)methyl)-2-(9-(pyridin-2-yl)-6-oxaspiro[4.5]decan-9-yl)ethanamin
(9R)-N-[(3-Methoxy-2-thienyl)methyl]-9-(2-pyridinyl)-6-oxaspiro[4.5]decane-9-ethanamine hydrochloride (1:1)
(R)-N-((3-Methoxythiophen-2-yl)methyl)-2-(9-(pyridin-2-yl)-6-oxaspiro[4.5]decan-9-yl)ethanamine hydrochloride
[(3-Methoxythiophen-2-yl)methyl]({2-[(9R)-9-(pyridin-2-yl)-6-oxaspiro-[4.5]decan-9-yl]ethyl})amine TRV-130 | [Molecular Formula]
C22H31ClN2O2S | [MDL Number]
MFCD28385856 | [MOL File]
1401031-39-7.mol | [Molecular Weight]
423.012 |
| Chemical Properties | Back Directory | [Melting point ]
White Solid | [storage temp. ]
Hygroscopic, -20°C Freezer, Under inert atmosphere | [solubility ]
DMSO (Slightly), Methanol (Slightly) | [form ]
Solid | [color ]
White to Light Brown | [Stability:]
Hygroscopic |
| Hazard Information | Back Directory | [Uses]
TRV-130 is a μ-opioid receptor (MOR) G protein-biased ligand. It is potently analgesic while causing less gastrointestinal dysfunction and respiratory suppression than morphine at equianalgesic doses. |
|
|