| Identification | Back Directory | [Name]
TELENZEPINE DIHYDROCHLORIDE | [CAS]
147416-96-4 | [Synonyms]
TelenzepineHydrochloride
Telenzepine dihydrochloide
TELENZEPINE DIHYDROCHLORIDE
JTQJFSQQHGPLOX-UHFFFAOYSA-N
Telenzepine hydrate dihydrochloride
TELENZEPINE DIHYDROCHLORIDE SELECTIVE M1 MUSCARIN
4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H)
4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H)thieno[3,4-b][1,5]benzodiazepin-10-onedihydrochloride
4,9-DIHYDRO-3-METHYL-4-[(4-METHYL-1-PIPERAZINYL)ACETYL]-10H-THIENO[3,4-B][1,5] BENZODIAZEPIN-10-ONE DIHYDROCHLORIDE | [Molecular Formula]
C19H22N4O2S | [MDL Number]
MFCD00083208 | [MOL File]
147416-96-4.mol | [Molecular Weight]
370.47 |
| Chemical Properties | Back Directory | [storage temp. ]
Store at RT | [solubility ]
H2O: >10 mg/mL
| [form ]
solid
| [color ]
white
| [Water Solubility ]
Soluble to 100 mM in water | [InChI]
1S/C19H22N4O2S.2ClH.H2O/c1-13-18-14(12-26-13)19(25)20-15-5-3-4-6-16(15)23(18)17(24)11-22-9-7-21(2)8-10-22;;;/h3-6,12H,7-11H2,1-2H3,(H,20,25);2*1H;1H2 | [InChIKey]
HZWCRPGARSMPNS-UHFFFAOYSA-N | [SMILES]
O.Cl.Cl.CN1CCN(CC1)CC(=O)N2c3ccccc3NC(=O)c4csc(C)c24 |
| Hazard Information | Back Directory | [Uses]
Antiulcerative;M1 muscarinic antagonist | [Biological Activity]
Selective high affinity muscarinic M 1 receptor antagonist (K i = 0.94 nM). Inhibits gastric acid secretion. | [Biochem/physiol Actions]
Telenzepine is an analog of pirenzepine and inhibits the secretion of gastric acid. It is an antagonist to M1-receptor and targets the oxyntic gastric glands and the salivary glands. | [storage]
Desiccate at RT |
|
| Company Name: |
Sigma-Aldrich
|
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021-61415566 800-8193336 |
| Website: |
https://www.sigmaaldrich.cn |
| Company Name: |
Energy Chemical
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| Tel: |
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| Website: |
http://www.energy-chemical.com |
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