| Identification | Back Directory | [Name]
N-Methyl-N-[[(1R)-1,2,3,4-tetrahydro-5-methoxy-1-naphthalenyl]methyl]-6-benzofuranethanamine mesylate | [CAS]
152148-64-6 | [Synonyms]
| [Molecular Formula]
C24H31NO5S | [MOL File]
152148-64-6.mol | [Molecular Weight]
445.57 |
| Hazard Information | Back Directory | [Description]
High affinityα2-adrenoceptor antagonist and selective 5-HT uptake inhibitor (Kivalues are 01 and 3.77 nM respectively). Displays low affinity at a variety of structurally homologous GPCRs. | [Uses]
A 80426 mesylate is an α2-adrenoceptor antagonist. A 80426 mesylate is used in antidepressant research[1]. | [IC 50]
α2-adrenergic receptor | [References]
[1] Hancock A A, et al. A‐80426, a potent α2‐adrenoceptor antagonist with serotonin uptake blocking activity and putative antidepressant‐like effects: I. Biochemical profile[J]. Drug Development Research, 1995, 35(4): 237-245. |
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BOC Sciences
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https://www.bocsci.com |
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