| Identification | Back Directory | [Name]
AC-ARG-PHE-MET-TRP-MET-ARG-NH2 | [CAS]
152274-65-2 | [Synonyms]
ACETALIN 1
AC-RFMWMR-NH2
OPIOID RECEPTOR ANTAGONIST 1
AC-ARG-PHE-MET-TRP-MET-ARG-NH2
L-Threoninamide,N2-acetyl-L-arginyl-L-phenylalanyl-L-methionyl-L-tryptophyl-L-methionyl
L-Threoninamide, N2-acetyl-L-arginyl-L-phenylalanyl-L-methionyl-L-tryptophyl-L-methionyl- (9CI) | [Molecular Formula]
C42H61N11O8S2 | [MDL Number]
MFCD00237472 | [MOL File]
152274-65-2.mol | [Molecular Weight]
912.13 |
| Hazard Information | Back Directory | [Uses]
Acetalin-3 (Ac-RFMWMT-NH2), a hexapeptide, is a μ opioid receptor antagonist with high affinity for μ and κ3 opioid receptor, weak affinity for κ1 receptors and no affinity for κ2 receptors[1]. | [IC 50]
μ Opioid Receptor/MOR | [References]
[1] C T Dooley, et al. Acetalins: opioid receptor antagonists determined through the use of synthetic peptide combinatorial libraries. Proc Natl Acad Sci U S A. 1993 Nov 15;90(22):10811-5. DOI:10.1073/pnas.90.22.10811 |
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