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1630083-70-3

1630083-70-3 Structure

1630083-70-3 Structure
IdentificationBack Directory
[Name]

E2027 maleate
[CAS]

1630083-70-3
[Synonyms]

E2027 maleate
Irsenontrine maleate
[Molecular Formula]

C26H26N4O7
[MOL File]

1630083-70-3.mol
[Molecular Weight]

506.52
Hazard InformationBack Directory
[Uses]

Irsenontrine (E2027) maleate is an orally active and selective phosphodiesterase 9 (PDE9) inhibitor. Irsenontrine maleate can be used for the research of neurological diseases[1][2].
[in vivo]

Irsenontrine (0.3, 3.3 mg/kg; p.o.) maleate exhibits a significant ameliorative effect on the percentage of exploration of the novel object at 3.3 mg/kg in Scopolamine-induced rats[1].
Irsenontrine (1 mg/kg; p.o.) maleate and memantine hydrochloride (1 mg/kg; p.o.) combined treatment group exhibits a significantly higher percentage of exploration of the novel object than memantine hydrochloride (1 mg/kg) alone[1].

[References]

[1] Miyamoto, et al. Dementia therapeutic agent combining pyrazoloquinoline derivative and memantine. WO2018221550 A1
[2] Hershey LA, et al. Pharmacological Management of Dementia with Lewy Bodies. Drugs Aging. 2019;36(4):309-319. DOI:10.1007/s40266-018-00636-7
[3] Eisai to present latest research on Alzheimer’s disease / dementia pipeline at the 14th international conference on Alzheimer’s & Parkinson’s diseases
1630083-70-3 suppliers list
Company Name: TargetMol Chemicals Inc.  
Tel: 15002134094
Website: https://www.targetmol.cn/
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