| Chemical Properties | Back Directory | [density ]
1.293±0.10 g/cm3(Temp: 25 °C; Press: 760 Torr)(predicted) | [form ]
Solid | [pka]
13.770±0.20(predicted) | [color ]
White to off-white |
| Hazard Information | Back Directory | [Uses]
BRD4 inhibitor-30 (Compound 1) is a BRD4 inhibitor with a IC50 value of 415 nM[1]. | [References]
[1] Koblan LW, et al. Assessment of Bromodomain Target Engagement by a Series of BI2536 Analogues with Miniaturized BET-BRET. ChemMedChem. 2016 Dec 6;11(23):2575-2581. DOI:10.1002/cmdc.201600502 |
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