| Identification | Back Directory | [Name]
Benzenebutanoic acid, 4-fluoro-β-[[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-2-[[(tricyclo[3.3.1.13,7]dec-2-yloxy)carbonyl]amino]propyl]amino]-, (βS)- | [CAS]
181941-32-2 | [Synonyms]
PD149164
PD-149164
PD 149164
Benzenebutanoic acid, 4-fluoro-β-[[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-2-[[(tricyclo[3.3.1.13,7]dec-2-yloxy)carbonyl]amino]propyl]amino]-, (βS)- | [Molecular Formula]
C33H38FN3O5 | [MOL File]
181941-32-2.mol | [Molecular Weight]
575.68 |
| Hazard Information | Back Directory | [Description]
PD-149164 is novel peptoid agonist for the CCK-A receptor. | [Uses]
PD-149164 is a potent agonist of cholecystokinin B (CCK-B) receptor, with IC50 values of 0.083 nM and 75 nM in binding assay to CCK-B and CCK-A[1]. | [IC 50]
CCKAR: 75 nM (IC50); CCKBR: 0.083 nM (IC50) | [References]
[1] J Hughes, et al. Characterization of novel peptoid agonists for the CCK-A receptor. Regul Pept. 1996 Aug 27;65(1):15-21. DOI:10.1016/0167-0115(96)00067-5 |
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