| Hazard Information | Back Directory | [Description]
YM 471 is an orally active, non-peptide arginine vasopressin (AVP) V1A and V2 receptor antagonist. | [Uses]
YM471 free base is a non-peptide antagonist of vasopressin V1A and V2 receptors with potent and persistent antagonistic activity. YM471 exhibits high affinity for rat V1A and V2 receptors with K values of 0.16 and 0.77 nM, respectively[1]. | [References]
[1] Pharmacological characterization of YM471, a novel potent vasopressin V(1A) and V(2) receptor antagonist DOI:10.1016/s0014-2999(02)01813-7 |
|
|