ChemicalBook--->CAS DataBase List--->2169946-15-8

2169946-15-8

2169946-15-8 Structure

2169946-15-8 Structure
IdentificationBack Directory
[Name]

Zanidatamab
[CAS]

2169946-15-8
[Synonyms]

Zanidatamab
Research Grade Zanidatamab
Research Grade Zanidatamab (DHC09607)
Chemical PropertiesBack Directory
[form ]

Liquid
[color ]

Colorless to light yellow
Hazard InformationBack Directory
[Uses]

Zanidatamab (ZW25) is a humanised, bispecific monoclonal antibody targeting 2 distinct HER2 epitopes (ECD2 and ECD4). Zanidatamab has anti-tumour activity[1].
[in vivo]

Zanidatamab (ZW25) induces significant tumor regressions, exhibiting 307% tumor growth inhibition relative to hIgG control and a 70% complete regression rate[1].

[IC 50]

HER2
[References]

[1] Weisser N, et, al. Preclinical development of a novel biparatopic HER2 antibody with activity in low to high HER2 expressing cancers. Cancer Res. 2017:77 (13).
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