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2543624-91-3

2543624-91-3 Structure

2543624-91-3 Structure
IdentificationBack Directory
[Name]

2-Amino-6-[4-(1,3-dihydro-1,3-dioxo-2H-isoindol-2-yl)phenyl]-4-(2-furanyl)-3-pyridinecarbonitrile
[CAS]

2543624-91-3
[Synonyms]

2-Amino-6-[4-(1,3-dihydro-1,3-dioxo-2H-isoindol-2-yl)phenyl]-4-(2-furanyl)-3-pyridinecarbonitrile
[Molecular Formula]

C24H14N4O3
[MOL File]

2543624-91-3.mol
[Molecular Weight]

406.39
Chemical PropertiesBack Directory
[Boiling point ]

678.4±65.0 °C(Predicted)
[density ]

1.50±0.1 g/cm3(Temp: 20 °C; Press: 760 Torr)(Predicted)
[pka]

3.24±0.18(Predicted)
Hazard InformationBack Directory
[Uses]

Pim-1 kinase inhibitor 2 (Compound 13) is a potent inhibitor of Pim-1 kinase. Pim-1 kinase inhibitor 2 induces apoptosis. Pim-1 kinase inhibitor 2 has the potential for the research of cancer diseases[1].
[References]

[1] Farrag AM, et al. New cyanopyridine-based scaffold as PIM-1 inhibitors and apoptotic inducers: Synthesis and SARs study. Bioorg Chem. 2020;105:104378. DOI:10.1016/j.bioorg.2020.104378
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