| Identification | Back Directory | [Name]
4H-Pyrrolo[3,2-c]pyridin-4-one, 1-[2-(2,4-difluorophenoxy)-5-[(ethylsulfonyl)methyl]-3-pyridinyl]-1,5-dihydro-3-methyl- | [CAS]
2760307-53-5 | [Synonyms]
BRD4 Inhibitor-23
4H-Pyrrolo[3,2-c]pyridin-4-one, 1-[2-(2,4-difluorophenoxy)-5-[(ethylsulfonyl)methyl]-3-pyridinyl]-1,5-dihydro-3-methyl- | [Molecular Formula]
C22H19F2N3O4S | [MOL File]
2760307-53-5.mol | [Molecular Weight]
459.47 |
| Hazard Information | Back Directory | [Uses]
BRD4 Inhibitor-23 is a potent and orally active BRD4 inhibitor with IC50s of 6.21 nM and 1.44 nM for BRD4 BD-1 and BRD4 BD-2, respectively (WO2022033542A1; Example 1)[1]. | [References]
[1] Chunli Shen, et al. 5-membered heteroaromatic pyridone compounds and application thereof. WO2022033542A1. |
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