| Identification | Back Directory | [Name]
(4BS,8R,8AS,14BR)-5,6,7,8,14,14B-HEXAHYDRO-7-(2-METHYL-2-PROPENYL)-4,8-METHANOBENZOFURO[2,3-A]PYRIDO[4,3-B]CARBAZOLE-1,8A(9H)-DIOL HYDROCHLORIDE | [CAS]
342884-62-2 | [Synonyms]
SDM25N
SDM25NHCl
SDM25N HYDROCHLORIDE
(4bS,8R,8aS,14bR)-5,6,7,8,14,14b-Hexahydro-7-(2-methyl-2-propenyl)-4,8-methanobenzofuro[2.3-a]pyrido[4.3-b]carbazole-1,8
4,8-Methanobenzofuro[2,3-a]pyrido[4,3-b]carbazole-1,8a(9H)-diol, 5,6,7,8,14,14b-hexahydro-7-(2-methyl-2-propen-1-yl)-, (4bS,8R,8aS,14bR)-
(4BS,8R,8AS,14BR)-5,6,7,8,14,14B-HEXAHYDRO-7-(2-METHYL-2-PROPENYL)-4,8-METHANOBENZOFURO[2,3-A]PYRIDO[4,3-B]CARBAZOLE-1,8A(9H)-DIOL HYDROCHLORIDE | [Molecular Formula]
C26H26N2O3 | [MDL Number]
MFCD06798365 | [MOL File]
342884-62-2.mol | [Molecular Weight]
414.5 |
| Chemical Properties | Back Directory | [Boiling point ]
630.5±55.0 °C(Predicted) | [density ]
1.44±0.1 g/cm3(Predicted) | [storage temp. ]
Store at +4°C | [solubility ]
DMSO: 2mg/mL, clear | [form ]
powder | [pka]
9.43±0.40(Predicted) | [color ]
white to beige |
| Hazard Information | Back Directory | [Biological Activity]
Potent and highly selective non-peptide δ receptor antagonist (K i values are 4.7, 3800 and 7900 nM for δ , κ and μ receptors respectively). More selective than naltrindole (17-(Cyclopropylmethyl)-6,7-dehydro-4,5a-epoxy-3,14-dihydroxy-6,7-2',3'-indolomorphinan hydrochloride ). |
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