| Identification | Back Directory | [Name]
PSB 1115 POTASSIUM SALT | [CAS]
409344-71-4 | [Synonyms]
PSB 1115
PSB-1115 (potassium)
PSB 1115 potassium salt hydrate
PSB 1115 hydrate potassium salt
1-Propyl-8-(4-sulfophenyl)xanthine potassium salt hydrate
1-Propyl-8-(4-sulfophenyl)xanthine hydrate potassium salt | [Molecular Formula]
C14H15KN4O5S | [MDL Number]
MFCD07784510 | [MOL File]
409344-71-4.mol | [Molecular Weight]
390.46 |
| Chemical Properties | Back Directory | [storage temp. ]
2-8°C | [solubility ]
DMSO: ~4 mg/mL | [form ]
solid | [color ]
off-white | [InChI]
1S/C14H14N4O5S.K/c1-2-7-18-13(19)10-12(17-14(18)20)16-11(15-10)8-3-5-9(6-4-8)24(21,22)23;/h3-6H,2,7H2,1H3,(H,15,16)(H,17,20)(H,21,22,23);/q;+1/p-1 | [InChIKey]
CJOWSBOERSTJAR-UHFFFAOYSA-M | [SMILES]
CCCN1C(=O)Nc2nc([nH]c2C1=O)-c3ccc(cc3)S(=O)(=O)O[K] |
| Hazard Information | Back Directory | [Uses]
PSB 1115 is an Adenosine A2B-R antagonist. | [Biological Activity]
Highly selective, water-soluble, human A 2B adenosine receptor antagonist. K i values are 53.4, > 10000 and > 10000 nM at human A 2B , A 1 and A 3 receptors respectively. Also selective versus rat A 1 and A 2A receptors (K i values are 2200 and 24000 nM respectively). Produces potent analgesic effects in vivo . | [Biochem/physiol Actions]
PSB 1115 is a highly selective, water-soluble, human A2B adenosine receptor antagonist. |
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| Company Name: |
Sigma-Aldrich
|
| Tel: |
021-61415566 800-8193336 |
| Website: |
https://www.sigmaaldrich.cn |
| Company Name: |
Merck KGaA
|
| Tel: |
21-20338288 |
| Website: |
www.sigmaaldrich.cn |
|