| Identification | Back Directory | [Name]
3-AMINO-N-[(4-CHLOROPHENYL)METHYL]-4,6-DIMETHYLTHIENO[2,3-B]PYRIDINE-2-CARBOXAMIDE | [CAS]
633283-39-3 | [Synonyms]
VU 10010
3-Amino-4,6-dimethyl-thieno[2,3-b]pyridine-2-carboxylic acid 4-chloro-benzylamide
3-AMINO-N-[(4-CHLOROPHENYL)METHYL]-4,6-DIMETHYLTHIENO[2,3-B]PYRIDINE-2-CARBOXAMIDE
Thieno[2,3-b]pyridine-2-carboxamide, 3-amino-N-[(4-chlorophenyl)methyl]-4,6-dimethyl- | [Molecular Formula]
C17H16ClN3OS | [MDL Number]
MFCD03821022 | [MOL File]
633283-39-3.mol | [Molecular Weight]
345.85 |
| Hazard Information | Back Directory | [Uses]
This compound acts as a selective allosteric M4 (Muscarinic Acetylcholine Receptor) agonist. | [Biological Activity]
Selective allosteric potentiator of M 4 acetylcholine receptors (EC 50 values are 33 and 0.7 nM for ACh in the absence and presence of VU10010 espectively). Binds to an allosteric site on the receptor increasing affinity for ACh and coupling to G-proteins. | [IC 50]
mAChR4 | [storage]
Store at -20°C |
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BOC Sciences
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https://www.bocsci.com |
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Energy Chemical
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021-58432009 400-005-6266 |
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http://www.energy-chemical.com |
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